Abstract
The 1,3-azole motif is a common and integral feature of many clinical drugs. Due to their wide-ranging applications, the development of 1,3-azoles as therapeutic agents is an ongoing focus of medicinal chemists. This review highlights the recent approaches towards the assembly of 1,3-oxazole, 1,3-thiazole and 1,3-imidazole motifs.
Keywords: 1, 3-Azoles, Imidazole, Oxazole, Synthesis, Therapeutic agent, Thiazole.
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Current Topics in Medicinal Chemistry
Title:Recent Advances in the Synthesis of 1,3-Azoles
Volume: 16 Issue: 30
Author(s): Nadale K. Downer-Riley and Yvette A. Jackson
Affiliation:
Keywords: 1, 3-Azoles, Imidazole, Oxazole, Synthesis, Therapeutic agent, Thiazole.
Abstract: The 1,3-azole motif is a common and integral feature of many clinical drugs. Due to their wide-ranging applications, the development of 1,3-azoles as therapeutic agents is an ongoing focus of medicinal chemists. This review highlights the recent approaches towards the assembly of 1,3-oxazole, 1,3-thiazole and 1,3-imidazole motifs.
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Cite this article as:
Downer-Riley K. Nadale and Jackson A. Yvette, Recent Advances in the Synthesis of 1,3-Azoles, Current Topics in Medicinal Chemistry 2016; 16 (30) . https://dx.doi.org/10.2174/1568026616666160414122349
DOI https://dx.doi.org/10.2174/1568026616666160414122349 |
Print ISSN 1568-0266 |
Publisher Name Bentham Science Publisher |
Online ISSN 1873-4294 |
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