Search Result "pyruvate kinase inhibitors"


Research Article

Flavonoids as Pyruvate Kinase M2 Inhibitor: An In silico Analysis

Journal: Letters in Drug Design & Discovery
Volume: 21 Issue: 13 Year: 2024 Page: 2661-2673
Author(s):

Research Article

Design, Synthesis, and Evaluation of Novel Pyruvate DehydrogenaseKinase Inhibitors

Journal: Medicinal Chemistry
Volume: 19 Issue: 3 Year: 2023 Page: 276-296
Author(s):

Therapeutic Potential of the Mammalian Pyruvate Dehydrogenase Kinases in the Prevention of Hyperglycaemia

Journal: Current Drug Targets - Immune, Endocrine & Metabolic Disorders
Volume: 2 Issue: 2 Year: 2002 Page: 151-165
Author(s): M. C. Sugden, M. J. Holness

Review Article

Inhibition of Pyruvate Dehydrogenase Kinase as a Therapeutic Strategy against Cancer

Journal: Current Topics in Medicinal Chemistry
Volume: 18 Issue: 6 Year: 2018 Page: 444-453
Author(s): Swatishree Sradhanjali,Mamatha M. Reddy

General Review Article

Methicillin-Resistant Staphylococcus Aureus (MRSA) Pyruvate Kinase(PK) Inhibitors and their Antimicrobial Activities

Journal: Current Medicinal Chemistry
Volume: 29 Issue: 5 Year: 2022 Page: 908-923
Author(s): Jingjing Jia,Yang Luo,Xue Zhong,Ling He

Research Article

Rationalization of the activity Profile of Pyruvate Kinase Isozyme M2 (PKM2) Inhibitors using 3D QSAR

Journal: Current Topics in Medicinal Chemistry
Volume: 21 Issue: 25 Year: 2021 Page: 2258-2271
Author(s): Merugumala Kusuma,Sahil Arora,Sourav Kalra,Anuhar Chaturvedi,Michael Heuser,Raj Kumar

Pyruvate Kinase M2: Regulatory Circuits and Potential for Therapeutic Intervention

Journal: Current Pharmaceutical Design
Volume: 20 Issue: 1 Year: 2014 Page: 2595-2606
Author(s): Vibhor Gupta, Kathryn E. Wellen, Sybille Mazurek, Rameshwar N. K. Bamezai

Pyruvate Dehydrogenase Kinases in the Nervous System: Their Principal Functions in Neuronal-glial Metabolic Interaction and Neuro-metabolic Disorders

Journal: Current Neuropharmacology
Volume: 10 Issue: 4 Year: 2012 Page: 393-403
Author(s): Mithilesh Kumar Jha,Sangmin Jeon,Kyoungho Suk

Small Molecule Kinase Inhibitors as Anti-Cancer Therapeutics

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 12 Issue: 5 Year: 2012 Page: 399-411
Author(s): O. Chahrour,D. Cairns,Z. Omran

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