Search Result "colchicine binding site"


Research Article

Structural Analysis for Colchicine Binding Site-Targeted ATCAA Derivatives as Melanoma Antagonists

Journal: Medicinal Chemistry
Volume: 10 Issue: 3 Year: 2014 Page: 277-286
Author(s): Jiawei Zhang,Feng Li,Yan Li,Yangyang Guo,Jinghui Wang,Shuwei Zhang

Review Article

Tubulin Inhibitors Binding to Colchicine-Site: A Review from 2015 to 2019

Journal: Current Medicinal Chemistry
Volume: 27 Issue: 40 Year: 2020 Page: 6787-6814
Author(s): Lin-Ying Xia,Ya-Liang Zhang,Rong Yang,Zhong-Chang Wang,Ya-Dong Lu,Bao-Zhong Wang,Hai-Liang Zhu

Current Frontiers

Butterfly Structure: A Privileged Scaffold Targeting Tubulin-Colchicine Binding Site

Journal: Current Topics in Medicinal Chemistry
Volume: 20 Issue: 17 Year: 2020 Page: 1505-1508
Author(s): Yingge Wang,Yongfang Yao,Hai-Liang Zhu,Yongtao Duan

Review Article

Recent Advances in Heterocyclic Tubulin Inhibitors Targeting the Colchicine Binding Site

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 16 Issue: 10 Year: 2016 Page: 1325-1338
Author(s): Xiaoxin Wu,Qinghui Wang,Wei Li

Recent Development and SAR Analysis of Colchicine Binding Site Inhibitors

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 9 Issue: 1 Year: 2009 Page: 1174-1190
Author(s): Jing Chen, Tao Liu, Xiaowu Dong, Yongzhou Hu

Pyridine Based Antitumour Compounds Acting at the Colchicine Site

Journal: Current Medicinal Chemistry
Volume: 23 Issue: 11 Year: 2016 Page: 1100-1130
Author(s): R. Álvarez,L. Aramburu,P. Puebla,E. Caballero,M. González,A. Vicente,M. Medarde,R. Peláez

Review Article

Targeting Tubulin-colchicine Site for Cancer Therapy: Inhibitors, Antibody- Drug Conjugates and Degradation Agents

Journal: Current Topics in Medicinal Chemistry
Volume: 19 Issue: 15 Year: 2019 Page: 1289-1304
Author(s): Yongtao Duan,Wei Liu,Liang Tian,Yanna Mao,Chuanjun Song

Tubulin Colchicine Binding Site Inhibitors as Vascular Disrupting Agents in Clinical Developments

Journal: Current Medicinal Chemistry
Volume: 22 Issue: 11 Year: 2015 Page: 1348-1360
Author(s): Ya-Ting Ji,Yan-Na Liu,Zhao-Peng Liu

New Ligands of the Tubulin Colchicine Site Based on X-Ray Structures

Journal: Current Topics in Medicinal Chemistry
Volume: 14 Issue: 20 Year: 2014 Page: 2231-2252
Author(s): Raquel Alvarez,Manuel Medarde,Rafael Pelaez

Research Article

Synthesis, Molecular Docking, and Biological Evaluation of 2,3-DiphenylquinoxalineDerivatives as a Tubulin’s Colchicine Binding Site Inhibitor Based on Primary VirtualScreening

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 22 Issue: 10 Year: 2022 Page: 2011-2025
Author(s): Massoud Amanlou,Mohsen Amini,Saeed Bahadorikhalili,Elnaz Rezaeiamiri,Mohammad Nazari Montazer,Mehdi Asadi,Zahra Rezaei

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