Search Result "estrone derivatives"
Synthesis, Biological Evaluation and the Rationalisation of the Inhibitory Activity of a Range of Sulfonate Derivatives of Estrone (E1) in the Design of Reversible Inhibitors of Estrone Sulfatase (ES)
Journal: Letters in Drug Design & Discovery
Volume: 11 Issue: 8 Year: 2014 Page: 985-992
Author(s): Mohsen Akbarzadeh,Timothy Cartledge,Sabbir Ahmed
Design and Synthesis of Two Chrysene Derivatives Using Estrone and Androsterone as Chemical Tools
Journal: Letters in Organic Chemistry
Volume: 13 Issue: 4 Year: 2016 Page: 237-248
Author(s): Lauro Figueroa-Valverde,Francisco DÃaz-Cedillo,Lenin Hau-Heredia,Marcela Rosas-Nexticapa,Benjamin Otto-Ortega,Elodia GarcÃa-Cervera,Eduardo Pool-Gómez,MarÃa López-Ramos
Steroidal δ-Alkenyl Oximes as Ambident Nucleophiles: Electrophile- Induced Formation of Oxazepane Derivatives in the Bis-Estrone Series
Journal: Letters in Organic Chemistry
Volume: 5 Issue: 1 Year: 2008 Page: 17-21
Author(s): Janos Wolfling, Erzsebet Mernyak, Zsolt Bikadi, Eszter Hazai, Laszlo Mark, Gyula Schneider
Homologation of Estrone or Estradiol. Appending a Carbon Substituent Into the 3-hydroxyestra-1,3,5-triene Skeleton
Journal: Current Organic Chemistry
Volume: 11 Issue: 4 Year: 2007 Page: 383-405
Author(s): S. Braune, S. Deb, T. Hase, K. Wahala
Structure-Activity Relationship Determination Study of a Series of Novel Compounds as Potential Inhibitors of the Enzyme Estrone Sulfatase (ES)
Journal: Letters in Drug Design & Discovery
Volume: 1 Issue: 1 Year: 2004 Page: 35-44
Author(s): Chirag K. Patel, Caroline P. Owen, Kwabina Aidoo-Gyamfi, Sabbir Ahmed
Synthesis and Biological Evaluation of a Range of Thiosemicarbazone - Based Compounds as Potential Inhibitors of Estrone Sulfatase (ES)
Journal: Letters in Drug Design & Discovery
Volume: 8 Issue: 3 Year: 2011 Page: 241-245
Author(s): Amit Kumar, Sukriti Singh, Hadi Bordbar, Timothy Cartledge, Sabbir Ahmed
Synthesis and Preliminary Biological Evaluation of Estrone Dimers
Journal: Letters in Drug Design & Discovery
Volume: 4 Issue: 3 Year: 2007 Page: 171-174
Author(s): Daniel Rabouina, Valerie Perrona, Blaise NZemba, Atul Guptaa, Rene-C. Gaudreault, Gervais Berube
Heterocyclization of Thiophenes Derived from Estrone Followed by Cytotoxic, HTRF Kinase and Pim-1 Kinase Evaluations
Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 18 Issue: 12 Year: 2018 Page: 1711-1728
Author(s): Mahmoud A. Abdelaziz Mahmoud,Rafat M. Mohareb,Meshari. A. Al-Sharif
Review of Estrone Sulfatase and its Inhibitors - An Important New Target Against Hormone Dependent Breast Cancer
Journal: Current Medicinal Chemistry
Volume: 9 Issue: 2 Year: 2002 Page: 263-273
Author(s): Sabbir Ahmed, Caroline P. Owen, Karen James, Luther Sampson, Chirag K. Patel
Synthesis and In Vitro Biochemical Evaluation of a Series of Cycloalkyl Esters of 4-Sulfamoylated Benzoic Acid as Inhibitors of Estrone Sulfatase (ES)
Journal: Letters in Drug Design & Discovery
Volume: 4 Issue: 6 Year: 2007 Page: 399-403
Author(s): Caroline P. Owen, Chirag K. Patel, Tim Cartledge, Sabbir Ahmed