Search Result "allosteric enhancer activity"


Allosteric Enhancers for A1 Adenosine Receptor

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 7 Issue: 6 Year: 2007 Page: 559-569
Author(s): Pier Giovanni Baraldi, Maria Antonietta Iaconinoto, Allan R. Moorman, Maria Dora Carrion, Carlota Lopez Cara, Delia Preti, Olga Cruz Lopez, Francesca Fruttarolo, Mojgan Aghazadeh Tabrizi, Romeo Romagnoli

A Common Molecular Motif Characterizes Extracellular Allosteric Enhancers of GPCR Aminergic Receptors and Suggests Enhancer Mechanism of Action

Journal: Current Medicinal Chemistry
Volume: 21 Issue: 32 Year: 2014 Page: 3673-3686
Author(s): Robert Root-Bernstein,Patrick F. Dillon

Allosteric Enhancers of A1 Adenosine Receptors: State of the Art and New Horizons for Drug Development

Journal: Current Medicinal Chemistry
Volume: 17 Issue: 3 Year: 2010 Page: 3488-3502
Author(s): R. Romagnoli, P. G. Baraldi, M. A. Tabrizi, S. Gessi, P. A. Borea, S. Merighi

Allosteric Drugs and Seven Transmembrane Receptors

Journal: Current Topics in Medicinal Chemistry
Volume: 13 Issue: 1 Year: 2013 Page: 5-13
Author(s): Terry Kenakin

Allosterism at Muscarinic Receptors: Ligands and Mechanisms

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 5 Issue: 6 Year: 2005 Page: 523-543
Author(s): N. J.M. Birdsall, S. Lazareno

Allosteric Modulation of Muscarinic Acetylcholine Receptors

Journal: Current Neuropharmacology
Volume: 5 Issue: 3 Year: 2007 Page: 157-167
Author(s): Karen J. Gregory, Patrick M. Sexton, Arthur Christopoulos

Allosteric Modulators for mGlu Receptors

Journal: Current Neuropharmacology
Volume: 5 Issue: 3 Year: 2007 Page: 187-194
Author(s): F. Gasparini, W. Spooren

Research Article

Medicinal Chemistry of P2X Receptors: Allosteric Modulators

Journal: Current Medicinal Chemistry
Volume: 22 Issue: 7 Year: 2015 Page: 929-941
Author(s): Christa E. Muller

Therapeutic Relevance of the Allosteric Modulation of the 5-HT Transporter

Journal: Current Signal Transduction Therapy
Volume: 4 Issue: 2 Year: 2009 Page: 82-87
Author(s): Ouissame Mnie-Filali, Mostafa El Mansari, Connie Sanchez, Nasser Haddjeri

Allosteric Modulators of the Human Calcium-Sensing Receptor:Structures, Sites of Action, and Therapeutic Potentials

Journal: Endocrine, Metabolic & Immune Disorders - Drug Targets
Volume: 8 Issue: 3 Year: 2008 Page: 192-197
Author(s): Jianxin Hu

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