Search Result "Estrone (E1)"
Synthesis, Biological Evaluation and the Rationalisation of the Inhibitory Activity of a Range of Sulfonate Derivatives of Estrone (E1) in the Design of Reversible Inhibitors of Estrone Sulfatase (ES)
Journal: Letters in Drug Design & Discovery
Volume: 11 Issue: 8 Year: 2014 Page: 985-992
Author(s): Mohsen Akbarzadeh,Timothy Cartledge,Sabbir Ahmed
Estrone (E1) Based Esters as Potential Inhibitors of Type 3 17β- hydroxysteroid Dehydrogenase (17β-HSD3) in the Treatment of Hormone-Dependent Prostate Cancer
Journal: Letters in Drug Design & Discovery
Volume: 7 Issue: 9 Year: 2010 Page: 650-656
Author(s): Moniola S. Olusanjo, Sabbir Ahmed
Synthesis, Biochemical Evaluation and Rationalisation of a Series of (3-O-Sulfonate) Derivatives of Estrone (E1) as Probes of the Active Site of Type 3 of the 17β-Hydroxysteroid Dehydrogenase (17β-HSD) Family of Enzymes
Journal: Letters in Drug Design & Discovery
Volume: 9 Issue: 1 Year: 2012 Page: 69-76
Author(s): Mohsen Akbarzadeh, Moniola S. Olusanjo, Sabbir Ahmed
Estrone Sulfatase and Its Inhibitors
Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 9 Issue: 6 Year: 2009 Page: 599-612
Author(s): Kwabina Aidoo-Gyamfi, Tim Cartledge, Kruti Shah, Sabbir Ahmed
Synthesis and Biological Evaluation of a Range of Thiosemicarbazone - Based Compounds as Potential Inhibitors of Estrone Sulfatase (ES)
Journal: Letters in Drug Design & Discovery
Volume: 8 Issue: 3 Year: 2011 Page: 241-245
Author(s): Amit Kumar, Sukriti Singh, Hadi Bordbar, Timothy Cartledge, Sabbir Ahmed
Review of Estrone Sulfatase and its Inhibitors - An Important New Target Against Hormone Dependent Breast Cancer
Journal: Current Medicinal Chemistry
Volume: 9 Issue: 2 Year: 2002 Page: 263-273
Author(s): Sabbir Ahmed, Caroline P. Owen, Karen James, Luther Sampson, Chirag K. Patel
Structure-Activity Relationship Determination Study of a Series of Novel Compounds as Potential Inhibitors of the Enzyme Estrone Sulfatase (ES)
Journal: Letters in Drug Design & Discovery
Volume: 1 Issue: 1 Year: 2004 Page: 35-44
Author(s): Chirag K. Patel, Caroline P. Owen, Kwabina Aidoo-Gyamfi, Sabbir Ahmed
Synthesis, In Vitro Activity and Rationalisation of a Series of Dialkyl Esters of 5-Aminosulfonylisophthanoate as Potential Estrone Sulfatase (ES) Inhibitors
Journal: Letters in Drug Design & Discovery
Volume: 11 Issue: 4 Year: 2014 Page: 437-443
Author(s): Sabbir Ahmed,Chirag K. Patel
Synthesis and In Vitro Biochemical Evaluation of a Series of Alkyl 6- Aminosulfonyl Naphthanoates as Potential Inhibitors of Human Placental Estrone Sulfatase (ES)
Journal: Letters in Drug Design & Discovery
Volume: 8 Issue: 1 Year: 2011 Page: 26-31
Author(s): Chirag K. Patel, Sabbir Ahmed
Chemical Synthesis, Characterisation and Biological Evaluation of Furanic- Estradiol Derivatives as Inhibitors of 17β-Hydroxysteroid Dehydrogenase Type 1
Journal: Medicinal Chemistry
Volume: 7 Issue: 2 Year: 2011 Page: 80-91
Author(s): Siham Farhane, Yannick Laplante, Donald Poirier