Search Result "DprE1"


Research Article

Identification of a Chemical Inhibitor with a Novel Scaffold TargetingDecaprenylphosphoryl-β-D-Ribose Oxidase (DprE1)

Journal: Infectious Disorders - Drug Targets
Volume: 23 Issue: 5 Year: 2023 Page: 24-30
Author(s):

DprE1 - from the Discovery to the Promising Tuberculosis Drug Target

Journal: Current Pharmaceutical Design
Volume: 20 Issue: 2 Year: 2014 Page: 4379-4403
Author(s): Katarina Miku sova, Vadim Makarov, Joao Neres

Computer-aided Identification of Novel DprE1 Inhibitors as Potential Anti-TB Lead Compounds: A Hybrid Virtual-screening and Molecular Dynamics Approach

Journal: Letters in Drug Design & Discovery
Volume: 12 Issue: 4 Year: 2015 Page: 302-313
Author(s): Yushir Maharaj,Soumendranath Bhakat,Mahmoud E. S. Soliman

Research Article

Antitubercular Potential of Novel Isoxazole Encompassed 1, 2, 4- Triazoles: Design, Synthesis, Molecular Docking Study and Evaluation of Antitubercular Activity

Journal: Anti-Infective Agents
Volume: 19 Issue: 2 Year: 2021 Page: 147-161
Author(s): Neenu Ganesh,Arun Kumar S,Manisha Singh,Venkaraddi Mangannavar Chandrashekar,Gurubasavaraj Veeranna Pujar

Decaprenylphosphoryl-β-D-Ribose 2-Epimerase from Mycobacterium tuberculosis is a Magic Drug Target

Journal: Current Medicinal Chemistry
Volume: 17 Issue: 2 Year: 2010 Page: 3099-3108
Author(s): G. Manina, M. R. Pasca, S. Buroni, E. De Rossi, G. Riccardi

Mini-Review Article

Selection of Suitable Protein Structure from Protein Data Bank: An ImportantStep in Structure-based Drug Design Studies

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 23 Issue: 3 Year: 2023 Page: 246-264
Author(s): Prashant R. Murumkar,Mayank Kumar Sharma,Niyati M. Patel,Mange Ram Yadav

Review Article

Exploring the Potential Inhibition of Candidate Drug Molecules for Clinical Investigation Based on their Docking or Crystallographic Analyses against M. tuberculosis Enzyme Targets

Journal: Current Topics in Medicinal Chemistry
Volume: 20 Issue: 29 Year: 2020 Page: 2662-2680
Author(s): Rishita Dey,Sisir Nandi,Asmita Samadder,Aaruni Saxena,Anil Kumar Saxena

Research Article

Synthesis, In-silico and In-vitro Antimycobacterial Studies on NovelBenzofuran Derivatives

Journal: Current Enzyme Inhibition
Volume: 19 Issue: 1 Year: 2023 Page: 2-9
Author(s): Dnyaneshwar E. Shelke,Bapu R. Thorat,Sanjay S. Dhabarde,Suraj N. Mali

Review Article

New and Old Hot Drug Targets in Tuberculosis

Journal: Current Medicinal Chemistry
Volume: 23 Issue: 33 Year: 2016 Page: 3813-3846
Author(s): Laurent Roberto Chiarelli,Giorgia Mori,Marta Esposito,Beatrice Silvia Orena,Maria Rosalia Pasca

Research Article

Novel Benzylidenehydrazide-1,2,3-Triazole Conjugates as Antitubercular Agents: Synthesis and Molecular Docking

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 19 Issue: 14 Year: 2019 Page: 1178-1194
Author(s): Mubarak H. Shaikh,Dnyaneshwar D. Subhedar,Laxman Nawale,Dhiman Sarkar,Firoz A. Kalam Khan,Jaiprakash N. Sangshetti,Bapurao B. Shingate

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