Search Result "2-aminothiazole hybrid"


Research Article

Biological Evaluation of 2-aminothiazole Hybrid as Antimalarial and Antitrypanosomal Agents: Design and Synthesis

Journal: Anti-Infective Agents
Volume: 18 Issue: 2 Year: 2020 Page: 101-108
Author(s): Surender S. Jadav,Vishnu N. Badavath,Ramesh Ganesan,Narayana M. Ganta,Dominique Besson,Venkatesan Jayaprakash

Research Article

Synthesis and Antitumor Activity Evaluation of 2-Aminothiazoles Appended 5-methylisoxazoline and Pyridine-piperazine Hybrid Molecules

Journal: Letters in Organic Chemistry
Volume: 15 Issue: 12 Year: 2018 Page: 1070-1077
Author(s): Garbapu Suresh,Ratnakaram Venkata Nadh,Navuluri Srinivasu,Durgaprasad Yennity

Review Article

Multitarget Tacrine Hybrids with Neuroprotective Properties to Confront Alzheimer's Disease

Journal: Current Topics in Medicinal Chemistry
Volume: 17 Issue: 9 Year: 2017 Page: 1006-1026
Author(s): Katarina Spilovska,Jan Korabecny,Eugenie Nepovimova,Rafael Dolezal,Eva Mezeiova,Ondrej Soukup,Kamil Kuca

Research Article

New Hybrids with 2-aminobenzothiazole and Azelayl Scaffolds: Synthesis, Molecular Docking and Biological Evaluation

Journal: Current Organic Chemistry
Volume: 22 Issue: 16 Year: 2018 Page: 1649-1660
Author(s): Carla Boga,Gabriele Micheletti,Isabel Orlando,Elena Strocchi,Beatrice Vitali,Laura Verardi,Giorgio Sartor,Natalia Calonghi

Recent Developments in the Third Generation Inhibitors of Bcr-Abl for Overriding T315I Mutation

Journal: Current Medicinal Chemistry
Volume: 18 Issue: 1 Year: 2011 Page: 2146-2157
Author(s): X. Y. Lu, Q. Cai, K. Ding

Research Article

Mechanochemical Synthesis, in vitro Evaluation and Molecular Docking Studies of 4-Amino-2-arylamino-5-(benzofuran-2-oyl)thiazoles as Antidiabetic Agents

Journal: Letters in Organic Chemistry
Volume: 16 Issue: 7 Year: 2019 Page: 560-568
Author(s): Vijayan R. Akhila,Maheswari R. Priya,Daisy R. Sherin,Girija K. Krishnapriya,Sreerekha V. Keerthi,Thanathu K. Manojkumar,Kallikat N. Rajasekharan

Review Article

Functionalized Morpholine-thiazole Scaffold: Synthetic Strategies andApplications

Journal: Current Organic Synthesis
Volume: 21 Issue: 6 Year: 2024 Page: 729-763
Author(s): Tarik E. Ali,Mohammed A. Assiri,Maha N. Alqahtani

Research Article

Identification of Degradation Products of Cefoselis Sulfate by HPLC-ESI-Quadrupole Time-Of-Flight-Mass Spectrometry in Aqueous Solutions

Journal: Current Pharmaceutical Analysis
Volume: 13 Issue: 1 Year: 2017 Page: 26-30
Author(s): Przemyslaw Zalewski,Robert Skibinski,Alicja Talaczynska,Magdalena Paczkowska,Judyta Cielecka-Piontek

Research Article

Development of Promising Thiopyrimidine-Based Anti-cancer and Antimicrobial Agents: Synthesis and QSAR Analysis

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 19 Issue: 15 Year: 2019 Page: 1255-1275
Author(s): Yasmin M. Syam,Manal M. Anwar,Eman R. Kotb,Samia A. Elseginy,Hanem M. Awad,Ghada E.A. Awad

Review Article

Thioureas as Building Blocks for the Generation of Heterocycles and Compounds with Pharmacological Activity: An Overview

Journal: Mini-Reviews in Organic Chemistry
Volume: 15 Issue: 1 Year: 2018 Page: 28-35
Author(s): Itamar Luís Goncalves,Gabriel Oliveira de Azambuja,Daniel Fabio Kawano,Vera Lucia Eifler-Lima

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