Search Result "bromodomain and extraterminal domain (BET) inhibitors"
Overexpression of Bromodomain and Extraterminal Domain is Associated withProgression, Metastasis and Unfavorable Outcomes: Highlighting Prognostic andTherapeutic Value of the BET Protein Family in Gastric Cancer
Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 23 Issue: 7 Year: 2023 Page: 794-806
Author(s): Shahrzad S. Fard,Seyed A. Mousavi,Seyed H. Ghaffari
Recent Advances in the Development of CBP/p300 Bromodomain Inhibitors
Journal: Current Medicinal Chemistry
Volume: 27 Issue: 33 Year: 2020 Page: 5583-5598
Author(s): Ying Xiong,Mingming Zhang,Yingxia Li
Prediction of Inhibition Activity of BET Bromodomain Inhibitors using Grid Search-Based Extreme Learning Machine and Molecular Docking
Journal: Letters in Drug Design & Discovery
Volume: 18 Issue: 11 Year: 2021 Page: 1039-1049
Author(s): Oluwatoba Emmanuel Oyeneyin,Babatunde Samuel Obadawo,Segun Michael Orimoloye,Eric Oluwafisayo Akintemi,Nureni Ipinloju,Adeola M. Asere,Taoreed O. Owolabi
Privileged Scaffolds Targeting Bromodomain-containing Protein 4
Journal: Current Topics in Medicinal Chemistry
Volume: 22 Issue: 7 Year: 2022 Page: 600-627
Author(s):
The Bromodomain and Extra-Terminal Protein Inhibitor OTX015 Suppresses T Helper Cell Proliferation and Differentiation
Journal: Current Molecular Medicine
Volume: 18 Issue: 9 Year: 2018 Page: 594-601
Author(s): Xiao Hu,Lauren P. Schewitz-Bowers,Philippa J. P. Lait,David A. Copland,Madeleine L. Stimpson,Jing Jing Li,Yizhi Liu,Andrew D. Dick,Richard W. J. Lee,Lai Wei
Aim for the Readers! Bromodomains As New Targets Against Chagas’ Disease
Journal: Current Medicinal Chemistry
Volume: 26 Issue: 3 Year: 2019 Page: 6544-6563
Author(s): Victoria Lucia Alonso,Luis Emilio Tavernelli,Alejandro Pezza,Pamela Cribb,Carla Ritagliati,Esteban Serra
Bromodomain Protein-directed Agents and MYC in Small Cell LungCancer
Journal: Current Cancer Drug Targets
Volume: 24 Issue: 9 Year: 2024 Page: 930-940
Author(s):
Piecing the Fragments Together: Dynamical Insights into the Enhancementof BRD4-BD1 (BET Protein) Druggability in Cancer ChemotherapyUsing Novel 8-methyl-pyrrolo[1,2-a]pyrazin-1(2H)-one Derivatives
Journal: Current Pharmaceutical Biotechnology
Volume: 23 Issue: 3 Year: 2022 Page: 444-456
Author(s): Oluwole B. Akawa,Opeyemi S. Soremekun,Fisayo A. Olotu,Mahmoud E.S. Solima
An Overview on Small Molecule Inhibitors of BRD4
Journal: Mini-Reviews in Medicinal Chemistry
Volume: 16 Issue: 17 Year: 2016 Page: 1403-1414
Author(s): Wenhai Huang,Xiaoliang Zheng,Yewei Yang,Xiaoju Wang,Zhengrong Shen
Targeting Epigenome As An Innovative Pharmacological Strategy For Castration-resistant Prostate Cancer
Journal: Clinical Cancer Drugs
Volume: 3 Issue: 1 Year: 2016 Page: 23-35
Author(s): Lavinia Casati, Fabio Celotti, Valeria Sibilia