Search Result "Dyrk1A"


DYRK1A Kinase Inhibitors with Emphasis on Cancer

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 12 Issue: 1 Year: 2012 Page: 1315-1329
Author(s): A. Ionescu, F. Dufrasne, M. Gelbcke, I. Jabin, R. Kiss, D. Lamoral-Theys

Review Article

DYRK1A Inhibitors and Perspectives for the Treatment of Alzheimer'sDisease

Journal: Current Medicinal Chemistry
Volume: 30 Issue: 6 Year: 2023 Page: 669-688
Author(s): Márcia Maria de Souza,Arthur Ribeiro Cenci,Kerolain Faoro Teixeira,Majory Christina Garcia Mendes Schuler,Ana Elisa Gonçalves,Leonardo Luiz Gomes Ferreira,Aldo Sena de Oliveira,Adriano Defini Andricopulo

DYRK1A: A Potential Drug Target for Multiple Down Syndrome Neuropathologies

Journal: CNS & Neurological Disorders - Drug Targets
Volume: 13 Issue: 1 Year: 2014 Page: 26-33
Author(s): Walter Becker,Ulf Soppa,Francisco J. Tejedor

Research Article

Overexpression of miR-26a-5p Suppresses Tau Phosphorylation and Aβ Accumulation in the Alzheimer’s Disease Mice by Targeting DYRK1A

Journal: Current Neurovascular Research
Volume: 17 Issue: 3 Year: 2020 Page: 241-248
Author(s): Yanni Liu,Lin Wang,Fuheng Xie,Xiao Wang,Yuanyuan Hou,Xiaomeng Wang,Juan Liu

QSAR and Pharmacophore Study of Dyrk1A Inhibitory Meridianin Analogs as Potential Agents for Treatment of Neurodegenerative Diseases

Journal: Medicinal Chemistry
Volume: 9 Issue: 1 Year: 2013 Page: 152-161
Author(s): Sandip B. Bharate, Rammohan R. Yadav, Ram A. Vishwakarma

Pharmacophore Based 3D-QSAR Modeling and Molecular Docking of Leucettines as Potent Dyrk1A Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 10 Issue: 8 Year: 2013 Page: 719-726
Author(s): Anu Bahl,Prashant Joshi,Sandip B. Bharate,Harish Chopra

Genetics of Down Syndrome: An Update

Ebook: Down Syndrome Children - An Update
Volume: 1 Year: 2015
Author(s): Solaf M. Elsayed
Doi: 10.2174/9781681081342115010005

Research Article

Design, Synthesis, Molecular Docking Study and Anti-Hepatocellular Carcinoma Evaluation of New Bis-Triazolothiadiazines

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 20 Issue: 9 Year: 2020 Page: 788-800
Author(s): Sobhi M. Gomha,Zeinab A. Muhammad,Elham Ezz El-Arab,Amira M. Elmetwally,Abdelaziz A. El-Sayed,Islam K. Matar

Regulation of Foxo-Dependent Transcription by Post-Translational Modifications

Journal: Current Drug Targets
Volume: 12 Issue: 9 Year: 2011 Page: 1303-1310
Author(s): Marco Boccitto, Robert G. Kalb

ATP Site-Directed Inhibitors of Protein Kinase CK2: An Update

Journal: Current Topics in Medicinal Chemistry
Volume: 11 Issue: 1 Year: 2011 Page: 1340-1351
Author(s): S. Sarno, E. Papinutto, C. Franchin, J. Bain, M. Elliott, F. Meggio, Z. Kazimierczuk, A. Orzeszko, G. Zanotti, R. Battistutta, L. A. Pinna

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