Search Result "Bromodomain-containing Protein 4 Bromodomain 1 (BRD4-BD1)"
Bromodomain-Containing Protein 4: A Druggable Target
Journal: Current Drug Targets
Volume: 20 Issue: 15 Year: 2019 Page: 1517-1536
Author(s): Yingying Shi,Jingwen Liu,Yuanyuan Zhao,Jiaoxian Cao,Yiming Li,Fujiang Guo
Privileged Scaffolds Targeting Bromodomain-containing Protein 4
Journal: Current Topics in Medicinal Chemistry
Volume: 22 Issue: 7 Year: 2022 Page: 600-627
Author(s):
Piecing the Fragments Together: Dynamical Insights into the Enhancementof BRD4-BD1 (BET Protein) Druggability in Cancer ChemotherapyUsing Novel 8-methyl-pyrrolo[1,2-a]pyrazin-1(2H)-one Derivatives
Journal: Current Pharmaceutical Biotechnology
Volume: 23 Issue: 3 Year: 2022 Page: 444-456
Author(s): Oluwole B. Akawa,Opeyemi S. Soremekun,Fisayo A. Olotu,Mahmoud E.S. Solima
Synthesis and Biological Activity of Quinoxalone Derivatives as BRD4 Bromodomain Inhibitors
Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 1 Year: 2017 Page: 50-57
Author(s): Bin Xu,Lei-Lei Zhao,Yi-Fei Yang,Jian Zhang,Ling-Yun Yang,Bing Zhang,Li Han,Hui-Bin Zhang,Jin-Pei Zhou
Prediction of Inhibition Activity of BET Bromodomain Inhibitors using Grid Search-Based Extreme Learning Machine and Molecular Docking
Journal: Letters in Drug Design & Discovery
Volume: 18 Issue: 11 Year: 2021 Page: 1039-1049
Author(s): Oluwatoba Emmanuel Oyeneyin,Babatunde Samuel Obadawo,Segun Michael Orimoloye,Eric Oluwafisayo Akintemi,Nureni Ipinloju,Adeola M. Asere,Taoreed O. Owolabi
Synthesis, Biological Evaluation and Molecular Docking Studies of Novel Trimethoxy-ring Derivatives as BRD4 Inhibitors
Journal: Letters in Drug Design & Discovery
Volume: 15 Issue: 1 Year: 2018 Page: 1319-1328
Author(s): Yan Yang,Zhiyi Yao
Small-Molecule BET Inhibitors in Clinical and Preclinical Development and Their Therapeutic Potential
Journal: Current Topics in Medicinal Chemistry
Volume: 15 Issue: 8 Year: 2015 Page: 776-794
Author(s): Lei Yu,Zhen Wang,Zhang Zhang,Xiaomei Ren,Xiaoyun Lu,Ke Ding
An Overview on Small Molecule Inhibitors of BRD4
Journal: Mini-Reviews in Medicinal Chemistry
Volume: 16 Issue: 17 Year: 2016 Page: 1403-1414
Author(s): Wenhai Huang,Xiaoliang Zheng,Yewei Yang,Xiaoju Wang,Zhengrong Shen
Dual-target Inhibitors Based on BRD4: Novel Therapeutic Approaches for Cancer
Journal: Current Medicinal Chemistry
Volume: 28 Issue: 9 Year: 2021 Page: 1775-1795
Author(s): Sitao Zhang,Yanzhao Chen,Chengsen Tian,Yujing He,Zeru Tian,Yichao Wan,Tingting Liu
Recent Advances in the Design and Development of Anticancer Molecules based on PROTAC Technology
Journal: Current Medicinal Chemistry
Volume: 28 Issue: 7 Year: 2021 Page: 1304-1327
Author(s): Zere Mukhamejanova,Yichen Tong,Qi Xiang,Fang Xu,Jiyan Pang