Search Result "BRD4 inhibitors"
An Overview on Small Molecule Inhibitors of BRD4
Journal: Mini-Reviews in Medicinal Chemistry
Volume: 16 Issue: 17 Year: 2016 Page: 1403-1414
Author(s): Wenhai Huang,Xiaoliang Zheng,Yewei Yang,Xiaoju Wang,Zhengrong Shen
Drug Discovery of Acetophenone Derivatives as BRD4 Inhibitors
Journal: Letters in Drug Design & Discovery
Volume: 17 Issue: 3 Year: 2020 Page: 323-329
Author(s): Zhimin Zhang,Wenhai Huang,Xiaoliang Zheng,Chuansheng Li,Zhengrong Shen
Dual-target Inhibitors Based on BRD4: Novel Therapeutic Approaches for Cancer
Journal: Current Medicinal Chemistry
Volume: 28 Issue: 9 Year: 2021 Page: 1775-1795
Author(s): Sitao Zhang,Yanzhao Chen,Chengsen Tian,Yujing He,Zeru Tian,Yichao Wan,Tingting Liu
Synthesis, Biological Evaluation and Molecular Docking Studies of Novel Trimethoxy-ring Derivatives as BRD4 Inhibitors
Journal: Letters in Drug Design & Discovery
Volume: 15 Issue: 1 Year: 2018 Page: 1319-1328
Author(s): Yan Yang,Zhiyi Yao
The Klf6 Super-enhancer Determines Klf6 Sensitivity to BRD4 Inhibitors in Human Hepatoma (HepG2) Cells
Journal: Current Biotechnology
Volume: 9 Issue: 3 Year: 2020 Page: 209-218
Author(s): KumChol Ri,MyongRyong Ri,YongJae Song,KyuHwan Kim,Chol Kim
Synthesis and Biological Activity of Quinoxalone Derivatives as BRD4 Bromodomain Inhibitors
Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 1 Year: 2017 Page: 50-57
Author(s): Bin Xu,Lei-Lei Zhao,Yi-Fei Yang,Jian Zhang,Ling-Yun Yang,Bing Zhang,Li Han,Hui-Bin Zhang,Jin-Pei Zhou
BRD4 Protein as a Target for Lung Cancer and Hematological CancerTherapy: A Review
Journal: Current Drug Targets
Volume: 24 Issue: 14 Year: 2023 Page: 1079-1092
Author(s):
Charting the Bromodomain BRD4: Towards the Identification of Novel Inhibitors with Molecular Similarity and Receptor Mapping
Journal: Letters in Drug Design & Discovery
Volume: 15 Issue: 9 Year: 2018 Page: 1002-1011
Author(s): Fernando D. Prieto-Martinez,Jose L. Medina-Franco
Bromodomain-Containing Protein 4: A Druggable Target
Journal: Current Drug Targets
Volume: 20 Issue: 15 Year: 2019 Page: 1517-1536
Author(s): Yingying Shi,Jingwen Liu,Yuanyuan Zhao,Jiaoxian Cao,Yiming Li,Fujiang Guo
Piecing the Fragments Together: Dynamical Insights into the Enhancementof BRD4-BD1 (BET Protein) Druggability in Cancer ChemotherapyUsing Novel 8-methyl-pyrrolo[1,2-a]pyrazin-1(2H)-one Derivatives
Journal: Current Pharmaceutical Biotechnology
Volume: 23 Issue: 3 Year: 2022 Page: 444-456
Author(s): Oluwole B. Akawa,Opeyemi S. Soremekun,Fisayo A. Olotu,Mahmoud E.S. Solima