Search Result "3H-pyrimidin-4-one"


Novel 2-hydrazino-pyrimidin-4(3H)-one Derivatives with Pseudofunctional- Similarity to Siderophores as Potential Antimycobacterial Agents

Journal: Medicinal Chemistry
Volume: 9 Issue: 1 Year: 2013 Page: 77-83
Author(s): Ranjeet Bairwa, Nilesh R. Tawari, Amruta Alate, Swapnil Anam, Mariam S. Degani, Muktikant Ray, Ramakrishna M. G. Rajan

Efficient Synthesis of 7-benzyl-5,6,7,8-tetrahydropyrido[4,3:4,5]thieno [2,3-d]pyrimidin-4(3H)-Ones Via Aza-Wittig Reaction

Journal: Letters in Organic Chemistry
Volume: 8 Issue: 9 Year: 2011 Page: 644-647
Author(s): Hong Chen, Kai Yan, Ming-Guo Liu

Design and Synthesis of 2-Methylthio-3-substituted-5,6-dimethylthieno [2,3-d] pyrimidin-4(3H)-ones as Analgesic, Anti-Inflammatory and Antibacterial Agents

Journal: Medicinal Chemistry
Volume: 3 Issue: 1 Year: 2007 Page: 67-73
Author(s): V. Alagarsamy, V. Raja Solomon, R. Meenac, K. V. Ramaseshu, K. Thirumurugan, S. Murugesan

Efficient Synthesis of Fused Pyrimidine Derivatives with Biological Activity via Aza-Wittig Reaction

Journal: Current Organic Synthesis
Volume: 8 Issue: 5 Year: 2011 Page: 752-763
Author(s): Ren Qingyun, Tan Xiaosong, He Hongwu

Research Article

Novel 1,2,3-Triazole-functionalized pyrido[3',2':4,5]furo[3,2-d]pyrimidin- 4(3H)-one Derivatives: Synthesis, Anticancer Activity, CoMFA and CoMSIA Studies

Journal: Letters in Organic Chemistry
Volume: 17 Issue: 12 Year: 2020 Page: 969-978
Author(s): Balakishan Vadla,Sailu Betala

Research Article

Synthesis and Molecular Docking of New Thiophene Derivatives as Lactate Dehydrogenase-A Inhibitors

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 19 Issue: 10 Year: 2019 Page: 833-841
Author(s): Abd El-Galil E. Amr,Mohamed F. El-Shehry,Alhussein A. Ibrahim,Hanaa M. Hosni,Mohamed A. Al-Omar,Hazem A. Ghabbour

Research Article

Synthesis and In Vitro Anticancer Activity of 6-Ferrocenylpyrimidin-4(3H)-one Derivatives

Journal: Current Organic Synthesis
Volume: 16 Issue: 1 Year: 2019 Page: 160-164
Author(s): Stanislav A. Grabovskiy,Rinat S. Muhammadiev,Lenar R. Valiullin,Ivan S. Raginov,Natalie N. Kabal'nova

CoMFA and CoMSIA 3D QSAR Models for a Series of Some Condensed Thieno[2,3-d]pyrimidin-4(3H)-ones with Antihistaminic (H1) Activity

Journal: Medicinal Chemistry
Volume: 9 Issue: 3 Year: 2013 Page: 389-401
Author(s): Meenakshi Singh,Sushil K. Singh,Mahesh T. Chhabria,Kamala Vasu,Dhaivat Pandya

Research Article

Synthesis of Novel 3(N,N-dialkylamino)alkyl/phenyl Substituted Thieno[2,3-d]pyrimidinones as H1-Anti-Histaminic and Antimicrobial Agents

Journal: Current Bioactive Compounds
Volume: 15 Issue: 1 Year: 2019 Page: 63-70
Author(s): Shiv Dev Singh,Arvind Kumar,Firoz Babar,Neetu Sachan,Arun Kumar Sharma

Research Article

Antihelminthic Activity of Some 2-Substituted Thieno[2,3-d]pyrimidin-4-ones

Journal: Letters in Drug Design & Discovery
Volume: 15 Issue: 8 Year: 2018 Page: 887-894
Author(s): Anelia Mavrova,Stefan Dimov,Dimitar Vuchev,Kameliya Anichina,Denitsa Yancheva

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