Search Result "transition state isosteres"
Targeting Enzymes with Phosphonate-Based Inhibitors: Mimics of Tetrahedral Transition States and Stable Isosteric Analogues of Phosphates
Journal: Current Enzyme Inhibition
Volume: 2 Issue: 1 Year: 2006 Page: 61-72
Author(s): L. Azema, R. Baron, S. Ladame
Inhibition of BACE-1 by Hydroxyethylsulfide, Hydroxyethylamine and Hydroxyethylurea Isosteric Replacements
Journal: Letters in Drug Design & Discovery
Volume: 2 Issue: 2 Year: 2005 Page: 109-112
Author(s): L. Rizzi, S. Romeo
Design, Synthesis and Docking Studies of Hydroxyethylamine and Hydroxyethylsulfide BACE-1 Inhibitors
Journal: Protein & Peptide Letters
Volume: 16 Issue: 1 Year: 2009 Page: 86-90
Author(s): Luca Rizzi, Nadia Vaiana, Francesca Sagui, Eva Genesio, Elena Pilli, Valentina Porcari, Sergio Romeo
Towards a Poly-Functional Synthetic-Antimalarial Vaccine: Incorporating Non-Natural Elements into Artificially-Made Peptides for Mimicking Functional Pathogen Ligand Structures Representing New Site-Directed Vaccine Components
Journal: Current Immunology Reviews (Discontinued)
Volume: 9 Issue: 4 Year: 2013 Page: 261-275
Author(s): Jose Manuel Lozano,Manuel Elkin Patarroyo
3,4-Dihydroxypyrrolidine as Glycosidase Inhibitor
Journal: Current Topics in Medicinal Chemistry
Volume: 9 Issue: 1 Year: 2009 Page: 34-57
Author(s): Katsuhiko Suzuki, Tatsuto Nakahara, Osamu Kanie
Computational Modeling of Coordination Chemistry of Transition Metal Cations in Zeolites and in Metal-organic Frameworks
Journal: Current Physical Chemistry
Volume: 2 Issue: 2 Year: 2012 Page: 189-199
Author(s): Hristiyan A. Aleksandrov, Petko St. Petkov, Georgi N. Vayssilov
Origin of Chiral Pharmacology Stereochemistry in Metalloprotease Inhibition
Journal: Mini-Reviews in Medicinal Chemistry
Volume: 1 Issue: 2 Year: 2001 Page: 155-161
Author(s): D. H. Kim
Recent Advances in the Synthesis and Applications of Reduced Amide Pseudopeptides
Journal: Current Medicinal Chemistry
Volume: 16 Issue: 1 Year: 2009 Page: 2289-2304
Author(s): Matej Zivec, Ziga Jakopin, Stanislav Gobec
Recent Progress in the Medicinal Chemistry of γ-Secretase Inhibitors
Journal: Current Topics in Medicinal Chemistry
Volume: 8 Issue: 1 Year: 2008 Page: 17-33
Author(s): Richard E. Olson, Charles F. Albright
New Cathepsin D Inhibitor Library Utilizing Hydroxyethyl Isosteres with Cyclic Tertiary Amines
Journal: Medicinal Chemistry
Volume: 8 Issue: 6 Year: 2012 Page: 1146-1154
Author(s): Rose M. McConnell, Kalyani Inapudi, Naveen Kadasala, Karthika Yarlagadda, Priya Velusamy, Matthew S. McConnell, Adam Green, Carol Trana, Kelley Sayyar, James S. McConnell