Search Result "estrone-3-O-sulfamate"
Structure-Activity Relationship Determination Study of a Series of Novel Compounds as Potential Inhibitors of the Enzyme Estrone Sulfatase (ES)
Journal: Letters in Drug Design & Discovery
Volume: 1 Issue: 1 Year: 2004 Page: 35-44
Author(s): Chirag K. Patel, Caroline P. Owen, Kwabina Aidoo-Gyamfi, Sabbir Ahmed
Synthesis and Biological Evaluation of a Range of Thiosemicarbazone - Based Compounds as Potential Inhibitors of Estrone Sulfatase (ES)
Journal: Letters in Drug Design & Discovery
Volume: 8 Issue: 3 Year: 2011 Page: 241-245
Author(s): Amit Kumar, Sukriti Singh, Hadi Bordbar, Timothy Cartledge, Sabbir Ahmed
Synthesis, Biological Evaluation and the Rationalisation of the Inhibitory Activity of a Range of Sulfonate Derivatives of Estrone (E1) in the Design of Reversible Inhibitors of Estrone Sulfatase (ES)
Journal: Letters in Drug Design & Discovery
Volume: 11 Issue: 8 Year: 2014 Page: 985-992
Author(s): Mohsen Akbarzadeh,Timothy Cartledge,Sabbir Ahmed
Recent Studies on Aromatase and Sulfatase Involved in Breast Cancer and their Inhibitors
Journal: Current Enzyme Inhibition
Volume: 16 Issue: 1 Year: 2020 Page: 20-44
Author(s): Subhajit Makar,Abhrajyoti Ghosh,Ashok Kumar,Sushil K. Singh
Review of Estrone Sulfatase and its Inhibitors - An Important New Target Against Hormone Dependent Breast Cancer
Journal: Current Medicinal Chemistry
Volume: 9 Issue: 2 Year: 2002 Page: 263-273
Author(s): Sabbir Ahmed, Caroline P. Owen, Karen James, Luther Sampson, Chirag K. Patel
Synthesis and In Vitro Biochemical Evaluation of a Series of Cycloalkyl Esters of 4-Sulfamoylated Benzoic Acid as Inhibitors of Estrone Sulfatase (ES)
Journal: Letters in Drug Design & Discovery
Volume: 4 Issue: 6 Year: 2007 Page: 399-403
Author(s): Caroline P. Owen, Chirag K. Patel, Tim Cartledge, Sabbir Ahmed
Molecular Modelling, Design, Synthesis and Biochemical Evaluation of a Range of Non-Steroidal Thiosemicarbazone-Based Inhibitors of Estrone Sulfatase (ES) - A Potential Insight into the Action of a Range of Allosteric Inhibitors of ES
Journal: Letters in Drug Design & Discovery
Volume: 8 Issue: 9 Year: 2011 Page: 889-896
Author(s): Amit Kumar, Sukriti Singh, Balkrishna Bhamare, Kruti Shah, Pallav S. Shah, Sabbir Ahmed
Synthesis, In Vitro Activity and Rationalisation of a Series of Dialkyl Esters of 5-Aminosulfonylisophthanoate as Potential Estrone Sulfatase (ES) Inhibitors
Journal: Letters in Drug Design & Discovery
Volume: 11 Issue: 4 Year: 2014 Page: 437-443
Author(s): Sabbir Ahmed,Chirag K. Patel
Synthesis and In Vitro Biochemical Evaluation of a Series of Alkyl 6- Aminosulfonyl Naphthanoates as Potential Inhibitors of Human Placental Estrone Sulfatase (ES)
Journal: Letters in Drug Design & Discovery
Volume: 8 Issue: 1 Year: 2011 Page: 26-31
Author(s): Chirag K. Patel, Sabbir Ahmed
Characterization of Carbonic Anhydrase Isozyme Specific Inhibition by Sulfamated 2-Ethylestra Compounds
Journal: Letters in Drug Design & Discovery
Volume: 8 Issue: 8 Year: 2011 Page: 678-684
Author(s): Katherine H. Sippel, Andre Stander, Chingkuang Tu, Balasubramanian Venkatakrishnan, Arthur H. Robbins, Mavis Agbandje-McKenna, Fourie Joubert, Annie M. Joubert, Robert McKenna