Search Result "Transactivation assay"
The Utility of Stable Cell Lines to Assess Species Differences in PXR Transactivation
Journal: Drug Metabolism Letters
Volume: 1 Issue: 2 Year: 2007 Page: 147-152
Author(s): Michael W. Sinz, Devin Pray, Judy Raucy
Transactivation Assays that Identify Indirect and Direct Activators of Human Pregnane X Receptor (PXR, NR1I2) and Constitutive Androstane Receptor (CAR, NR1I3)
Journal: Drug Metabolism Letters
Volume: 11 Issue: 2 Year: 2017 Page: 128-137
Author(s): Marija Pinne,Elsa Ponce,Judy L. Raucy
Evaluation of 170 Xenobiotics as Transactivators of Human Pregnane X Receptor (hPXR) and Correlation to Known CYP3A4 Drug Interactions
Journal: Current Drug Metabolism
Volume: 7 Issue: 4 Year: 2006 Page: 375-388
Author(s): Michael Sinz, Sean Kim, Zhengrong Zhu, Taosheng Chen, Monique Anthony, Kenneth Dickinson, A. D. Rodrigues
Therapeutic Targeting of G-Protein Coupled Receptor-Mediated Epidermal Growth Factor Receptor Transactivation in Human Glioma Brain Tumors
Journal: Mini-Reviews in Medicinal Chemistry
Volume: 8 Issue: 1 Year: 2008 Page: 1418-1428
Author(s): M. Paolillo, S. Schinelli
Development of a Novel Reporter Gene Vector for Cell Based Angiogenic Studies
Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 14 Issue: 8 Year: 2011 Page: 703-709
Author(s): Srinivasan Kokatam, Deepshikha Pandey, Ramkrishna Gupta, Rathu Krishna, Rajeev Soni
Effect of Stilbene and Chalcone Scaffolds Incorporation in Clofibric Acid on PPARα Agonistic Activity
Journal: Medicinal Chemistry
Volume: 10 Issue: 1 Year: 2014 Page: 59-65
Author(s):
HIV-1 Infected Patients have Antibodies Recognizing Folded Tat
Journal: Infectious Disorders - Drug Targets
Volume: 11 Issue: 1 Year: 2011 Page: 57-63
Author(s): Sonia Mediouni, Gilbert Baillat, Albert Darque, Isabelle Ravaux, Erwann Loret
Miniaturization of a Panel of High Throughput Yeast-Cell-Based Nuclear Receptor Assays in 384- and 1536-Well Microplates
Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 14 Issue: 1 Year: 2011 Page: 47-54
Author(s): Johanna Rajasarkka, Marko Virta
Synthesis and Biological Evaluation of Gemfibrozil Chiral Analogues as Potential PPARα Agonists
Journal: Letters in Drug Design & Discovery
Volume: 8 Issue: 2 Year: 2011 Page: 154-158
Author(s): Barbara De Filippis, Letizia Giampietro, Antonella Giancristofaro, Alessandra Ammazzalorso, Marialuigia Fantacuzzi, Cristina Maccallini, Michele Petruzzelli, Rosa Amoroso
High-Throughput Screening Assays to Discover Small-Molecule Inhibitors of Protein Interactions
Journal: Current Drug Discovery Technologies
Volume: 5 Issue: 3 Year: 2008 Page: 190-199
Author(s): Pierre Colas