Abstract
This report deals with our recent results concerning the reaction and synthetic application of boronsubstituted heteroaromatic compounds (1) palladium-catalyzed cross-coupling, carbonylative cross-coupling and tandem cyclization cross-coupling reactions with dialkylpyridylboranes and indolylborates, and their use in the preparation of heterocyclic derivatives and (2) the synthetic application of an intramolecular alkyl migration process in indolylborates for the construction of more elaborate indole derivatives.
Keywords: heteroarylboron compound, indole derivatives, tandem cyclizaation
Call for Papers in Thematic Issues
Catalytic C-H bond activation as a tool for functionalization of heterocycles
The major topic is the functionalization of heterocycles through catalyzed C-H bond activation. The strategies based on C-H activation not only provide straightforward formation of C-C or C-X bonds but, more importantly, allow for the avoidance of pre-functionalization of one or two of the cross-coupling partners. The beneficial impact of ...read more
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