Search Result "thymidine"


Thymidine Phosphorylase Inhibitors

Ebook: Anti-Angiogenesis Drug Discovery and Development
Volume: 1 Year: 2011
Author(s): Radim Nencka
Doi: 10.2174/978160805162511101010116

N3-Substituted Thymidine Analogues: Radiosyntheses of N3-[4-(4-(2-[18F] fluoroethyl)phenyl)butyl]thymidine and N3-[5-(4-(2-[18F]fluoroethyl)- phenyl)pentyl]thymidine for PET

Journal: Current Radiopharmaceuticals
Volume: 2 Issue: 1 Year: 2009 Page: 2-8
Author(s): Pradip Ghosh, Juri G. Gelovani, Mian M. Alauddin

Synthesis of N3-Substituted Thymidine Analogues for Measurement of Cellular Kinase Activity

Journal: Medicinal Chemistry
Volume: 4 Issue: 5 Year: 2008 Page: 503-512
Author(s): P. Ghosh, A. Pal, A. Shavrin, W. Bornmann, J. G. Gelovani, M. M. Alauddin

Mitochondrial Thymidine Kinase Inhibitors

Journal: Current Topics in Medicinal Chemistry
Volume: 5 Issue: 1 Year: 2005 Page: 1205-1219
Author(s): Maria-Jesus Perez-Perez, Ana-Isabel Hernandez, Eva-Maria Priego, Fatima Rodriguez-Barrios, Federico Gago, Maria-Jose Camarasa, Jan Balzarini

The Role of Thymidine Kinases in the Activation of Pyrimidine Nucleoside Analogues

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 4 Issue: 4 Year: 2004 Page: 341-350
Author(s): Ashraf S. Al-Madhoun, Werner Tjarks, Staffan Eriksson

Role of Thymidine Phosphorylase in Biomodulation of Fluoropyrimidines

Journal: Current Pharmaceutical Biotechnology
Volume: 2 Issue: 3 Year: 2001 Page: 257-267
Author(s): T. Morita, A. Matsuzaki, K. Suzuki, A. Tokue

CycloSal-dRFIB, a Thymidine Mimetic, Thymidine Kinase by-Pass Nucleoside Prodrug: Radioiodination, in vitro Cellular Uptake and Biodistribution in Murine Models

Journal: Current Radiopharmaceuticals
Volume: 3 Issue: 4 Year: 2010 Page: 267-274
Author(s): Anke Stahlschmidt, William Sun, Aihua Zhou, Hans- Jurgen Machulla, Edward E. Knaus, Leonard I. Wiebe

Thymidine Phosphorylase and Fluoropyrimidines Efficacy: A Jekyl and Hyde Story

Journal: Current Medicinal Chemistry - Anti-Cancer Agents
Volume: 4 Issue: 2 Year: 2004 Page: 71-81
Author(s): Joseph Ciccolini, Alexandre Evrard, Pierre Cuq

Review Article

Exploring Pyrimidine Pharmacophore as Thymidine Monophosphate Kinase Inhibitors for Antitubercular Activity: A Review

Journal: Current Topics in Medicinal Chemistry
Volume: 16 Issue: 28 Year: 2016 Page: 3211-3223
Author(s): Trupti Sameer Chitre,Kalyani Dhirendra Asgaonkar,Shital Manoj Patil,Muthu Kumaradoss Kathiravan,Subhash Balkrishna Padhye

Thymidine Phosphorylase/Platelet-Derived Endothelial Cell Growth Factor as a Target for Capecitabine: From Biology to the Bedsid

Ebook: Frontiers in Anti-Cancer Drug Discovery
Volume: 1 Year: 2010
Author(s): Girolamo Ranieri, Aldo Maria Roccaro, Angelo Vacca, Domenico Ribatti
Doi: 10.2174/978160805161811001010031

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