Search Result "prediction model for CNS permeability"


Review Article

Blood Brain Barrier Permeability Prediction Using Machine Learning Techniques: An Update

Journal: Current Pharmaceutical Biotechnology
Volume: 20 Issue: 14 Year: 2019 Page: 1163-1171
Author(s): Deeksha Saxena,Anju Sharma,Mohammed H. Siddiqui,Rajnish Kumar

Patented In Vitro Blood-Brain Barrier Models in CNS Drug Discovery

Journal: Recent Patents on CNS Drug Discovery (Discontinued)
Volume: 6 Issue: 2 Year: 2011 Page: 107-118
Author(s): Andrea Toth, Szilvia Veszelka, Shinsuke Nakagawa, Masami Niwa, Maria A. Deli

In Silico Prediction Models for Blood-Brain Barrier Permeation

Journal: Current Medicinal Chemistry
Volume: 11 Issue: 1 Year: 2004 Page: 1617-1628
Author(s): Gerhard F. Ecker, Christian R. Noe

Research Article

Development of Machine Learning Based Blood-brain Barrier Permeability Prediction Models Using Physicochemical Properties, MACCS and Substructure Fingerprints

Journal: Current Bioinformatics
Volume: 16 Issue: 6 Year: 2021 Page: 855-864
Author(s): Deeksha Saxena,Anju Sharma,Mohammed Haris Siddiqui,Rajnish Kumar

Role of Microfluidics in Blood-Brain Barrier Permeability Cell Culture Modeling: Relevance to CNS Disorders

Journal: CNS & Neurological Disorders - Drug Targets
Volume: 15 Issue: 3 Year: 2016 Page: 301-309
Author(s): Alexander L. Rusanov,Natalia G. Luzgina,George E. Barreto,Gjumrakch Aliev

Review Article

Current State and Future Perspectives in QSAR Models to Predict Blood- Brain Barrier Penetration in Central Nervous System Drug R&D

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 17 Issue: 3 Year: 2017 Page: 247-257
Author(s): Juan F. Morales,Sebastian Scioli Montoto,Pietro Fagiolino,Maria E. Ruiz

Solubility and Permeability Measurement and Applications in Drug Discovery

Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 13 Issue: 2 Year: 2010 Page: 101-111
Author(s): Philip S. Burton, Jay T. Goodwin

CNS Drug Development – Lost in Translation?

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 12 Issue: 10 Year: 2012 Page: 959-970
Author(s): A. Talevi,C. L. Bellera,M. Di Ianni,M. Gantner,L. E. Bruno-Blanch,. A. Castro

Hurdles with Using In Vitro Models to Predict Human Blood-brain Barrier Drug Permeability: A Special Focus on Transporters and Metabolizing Enzymes

Journal: Current Drug Metabolism
Volume: 14 Issue: 1 Year: 2013 Page: 120-136
Author(s): Ramzi Shawahna,Xavier Decleves,Jean-Michel Scherrmann

Computational Models for Central Nervous System Penetration

Journal: Current Computer-Aided Drug Design
Volume: 5 Issue: 2 Year: 2009 Page: 71-89
Author(s): Anthony E. Klon

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