Search Result "hERG screening"
A Ligand-Based Virtual Screening Approach to Identify Small Molecules as hERG Channel Activators
Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 18 Issue: 3 Year: 2015 Page: 269-280
Author(s): Elisa Giacomini,Rosa Buonfiglio,Matteo Masetti,Yuhong Wang,Gea-Ny Tseng,Marinella Roberti,Maurizio Recanatini
Ligand Structural Aspects of hERG Channel Blockade
Journal: Current Topics in Medicinal Chemistry
Volume: 8 Issue: 1 Year: 2008 Page: 1113-1127
Author(s): Alex M. Aronov
Tuning hERG Out: Antitarget QSAR Models for Drug Development
Journal: Current Topics in Medicinal Chemistry
Volume: 14 Issue: 11 Year: 2014 Page: 1399-1415
Author(s): Rodolpho C. Braga,Vinicius M. Alves,Meryck F.B. Silva,Eugene Muratov,Denis Fourches,Alexander Tropsha,Carolina H. Andrade
hERG (KCNH2 or Kv11.1) K+ Channels: Screening for Cardiac Arrhythmia Risk
Journal: Current Drug Metabolism
Volume: 9 Issue: 9 Year: 2008 Page: 965-970
Author(s): Mark R. Bowlby, Ravi Peri, Howard Zhang, John Dunlop
In Silico hERG Modeling: Challenges and Progress
Journal: Current Computer-Aided Drug Design
Volume: 5 Issue: 2 Year: 2009 Page: 106-121
Author(s): David J. Diller
Recent Developments in Computational Prediction of hERG Blockage
Journal: Current Topics in Medicinal Chemistry
Volume: 13 Issue: 11 Year: 2013 Page: 1317-1326
Author(s): Sichao Wang,Youyong Li,Lei Xu,Dan Li,Tingjun Hou
How to Fluorescently Label the Potassium Channel: A Case in hERG
Journal: Current Medicinal Chemistry
Volume: 27 Issue: 18 Year: 2020 Page: 3046-3054
Author(s): Xiaomeng Zhang,Beilei Wang,Zhenzhen Liu,Yubin Zhou,Lupei Du
The hERG Channel and Risk of Drug-Acquired Cardiac Arrhythmia: An Overview
Journal: Current Topics in Medicinal Chemistry
Volume: 8 Issue: 1 Year: 2008 Page: 1102-1112
Author(s): Armando A. Lagrutta, Elena S. Trepakova, Joseph J. Salata
Lead Optimization of Melanin Concentrating Hormone Receptor 1 Antagonists with low hERG Channel Activity
Journal: Current Topics in Medicinal Chemistry
Volume: 8 Issue: 1 Year: 2008 Page: 1152-1157
Author(s): Andrew S. Judd, Andrew J. Souers, Philip R. Kym
Overcoming hERG Affinity in the Discovery of Maraviroc; A CCR5 Antagonist for the Treatment of HIV
Journal: Current Topics in Medicinal Chemistry
Volume: 8 Issue: 1 Year: 2008 Page: 1140-1151
Author(s): David A. Price, Duncan Armour, Marcel de Groot, Derek Leishman, Carolyn Napier, Manos Perros, Blanda L. Stammen, Anthony Wood