Search Result "crystallographic assay"
Elaboration of Novel TTK1 Inhibitory Leads via QSAR-Guided Selection of Crystallographic Pharmacophores Followed By In Vitro Assay
Journal: Current Computer-Aided Drug Design
Volume: 17 Issue: 4 Year: 2021 Page: 511-522
Author(s): Mahmoud A. Al-Sha'er,Mutasem O. Taha
Kinetic and Crystallographic Studies on Glyceraldehyde-3-Phosphate Dehydrogenase from Trypanosoma cruzi in Complex with Iodoacetate
Journal: Letters in Drug Design & Discovery
Volume: 6 Issue: 3 Year: 2009 Page: 210-214
Author(s): Rafael V.C. Guido, Tatiane L. Balliano, Adriano D. Andricopulo, Glaucius Oliva
Structural Insight Into the Crucial Role of Ligand Chirality in the Activation of PPARs by Crystallographic Methods
Journal: Current Topics in Medicinal Chemistry
Volume: 11 Issue: 7 Year: 2011 Page: 819-839
Author(s): F. Loiodice, G. Pochetti
Cross-Neutralizing Human Monoclonal Anti-HIV-1 Antibody 2F5: Preparation and Crystallographic Analysis of the Free and Epitope-Complexed Forms of its F ab Fragment
Journal: Protein & Peptide Letters
Volume: 8 Issue: 5 Year: 2001 Page: 413-418
Author(s): Steve Bryson, Annie Cunningham, Jason Ho, Rosemary C. Hynes, David E. Isenman, Brian H. Barber, Renate Kunert, Hermann Katinger, Michel Klein, Emil F. Pai
Identification, Characterization and Molecular Modelling Studies of Schistosoma mansoni Dihydrofolate Reductase Inhibitors: From Assay Development to Hit Identification
Journal: Current Topics in Medicinal Chemistry
Volume: 18 Issue: 5 Year: 2018 Page: 406-417
Author(s): Andre Lacerda Braga Teles,Roseane R. Silva,Michelle Ko,Glaucio Monteiro Ferreira,Samuel da Rocha Pita,Gustavo Henrique Goulart Trossini,Paulo Carvalho,Marcelo Santos Castilho
Lipophilic Mediated Assays for β-Hematin Inhibitors
Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 13 Issue: 3 Year: 2010 Page: 285-292
Author(s): Melissa D. Carter, Vanessa V. Phelan, Rebecca D. Sandlin, Brian O. Bachmann, David W. Wright
NMR Applications for Identifying β-TrCP Protein-Ligand Interactions
Journal: Mini-Reviews in Medicinal Chemistry
Volume: 11 Issue: 4 Year: 2011 Page: 283-297
Author(s): J. Pons, V. Tanchou, J.-P. Girault, G. Bertho, N. Evrard-Todeschi
A High Throughput Fluorescence Polarization Assay for Inhibitors of the GoLoco Motif/G-alpha Interaction
Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 11 Issue: 5 Year: 2008 Page: 396-409
Author(s): Adam J. Kimple, Adam Yasgar, Mark Hughes, Ajit Jadhav, Francis S. Willard, Robin E. Muller, Christopher P. Austin, James Inglese, Gordon C. Ibeanu, David P. Siderovski, Anton Simeonov
Crystallographic Study and Biological Evaluation of 1,4-dimethyl-N-alkylcarbazoles†
Journal: Current Topics in Medicinal Chemistry
Volume: 15 Issue: 11 Year: 2015 Page: 973-979
Author(s): Carmela Saturnino,Anna Caruso,Pasquale Longo,Anna Capasso,Attilio Pingitore,Maria Cristina Caroleo,Erika Cione,Mariarita Perri,Francesco Nicolo,Viviana Mollica Nardo,Luigi Monsu Scolaro,Maria Stefania Sinicropi,Maria Rosaria Plutino,Hussein El-Kashef
Preliminary X-Ray Crystallographic Studies Of The Mycobacterium Tuberculosis Hsp16.3 Molecular Chaperone
Journal: Protein & Peptide Letters
Volume: 8 Issue: 6 Year: 2001 Page: 499-502
Author(s): Y. Chen, J. An, Y. Ding, H. Dai, Q. Mao, L. Feng, B. Liu, Y. Chang, F. Chen, H. He, H. Tang, Z. Chang, Z. Rao