Search Result "blockers and activators of hERG"
The Interactions Between hERG Potassium Channel and Blockers
Journal: Current Topics in Medicinal Chemistry
Volume: 9 Issue: 4 Year: 2009 Page: 330-338
Author(s): Lupei Du, Minyong Li, Qidong You
Recent Developments in Computational Prediction of hERG Blockage
Journal: Current Topics in Medicinal Chemistry
Volume: 13 Issue: 11 Year: 2013 Page: 1317-1326
Author(s): Sichao Wang,Youyong Li,Lei Xu,Dan Li,Tingjun Hou
Tuning hERG Out: Antitarget QSAR Models for Drug Development
Journal: Current Topics in Medicinal Chemistry
Volume: 14 Issue: 11 Year: 2014 Page: 1399-1415
Author(s): Rodolpho C. Braga,Vinicius M. Alves,Meryck F.B. Silva,Eugene Muratov,Denis Fourches,Alexander Tropsha,Carolina H. Andrade
Ligand Structural Aspects of hERG Channel Blockade
Journal: Current Topics in Medicinal Chemistry
Volume: 8 Issue: 1 Year: 2008 Page: 1113-1127
Author(s): Alex M. Aronov
In Silico Predictions of hERG Channel Blockers in Drug Discovery: From Ligand-Based and Target-Based Approaches to Systems Chemical Biology
Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 14 Issue: 5 Year: 2011 Page: 375-387
Author(s): Olivier Taboureau, Flemming Steen Jorgensen
Implications of Dynamic Occupancy, Binding Kinetics, and Channel Gating Kinetics for hERG Blocker Safety Assessment and Mitigation
Journal: Current Topics in Medicinal Chemistry
Volume: 16 Issue: 16 Year: 2016 Page: 1792-1818
Author(s): Robert A. Pearlstein,K. Andrew MacCannell,Gül Erdemli,Sarita Yeola,Gabriel Helmlinger,Qi-Ying Hu,Ramy Farid,William Egan,Steven Whitebread,Clayton Springer,Jeremy Beck,Hao-Ran Wang,Mateusz Maciejewski,Laszlo Urban,José S. Duca
In Silico hERG Modeling: Challenges and Progress
Journal: Current Computer-Aided Drug Design
Volume: 5 Issue: 2 Year: 2009 Page: 106-121
Author(s): David J. Diller
QSAR and Pharmacophore Analysis of a Series of Piperidinyl Urea Derivatives as hERG Blockers and H3 Antagonists
Journal: Current Drug Discovery Technologies
Volume: 10 Issue: 1 Year: 2013 Page: 47-58
Author(s): N. S. Hari Narayana Moorthy, Maria J. Ramos, Pedro A. Fernandes
hERG (KCNH2 or Kv11.1) K+ Channels: Screening for Cardiac Arrhythmia Risk
Journal: Current Drug Metabolism
Volume: 9 Issue: 9 Year: 2008 Page: 965-970
Author(s): Mark R. Bowlby, Ravi Peri, Howard Zhang, John Dunlop
How to Fluorescently Label the Potassium Channel: A Case in hERG
Journal: Current Medicinal Chemistry
Volume: 27 Issue: 18 Year: 2020 Page: 3046-3054
Author(s): Xiaomeng Zhang,Beilei Wang,Zhenzhen Liu,Yubin Zhou,Lupei Du