Search Result "PKM2 inhibitors"


General Review Article

Recent Advances on PKM2 Inhibitors and Activators in CancerApplications

Journal: Current Medicinal Chemistry
Volume: 31 Issue: 20 Year: 2024 Page: 2955-2973
Author(s):

Research Article

Rationalization of the activity Profile of Pyruvate Kinase Isozyme M2 (PKM2) Inhibitors using 3D QSAR

Journal: Current Topics in Medicinal Chemistry
Volume: 21 Issue: 25 Year: 2021 Page: 2258-2271
Author(s): Merugumala Kusuma,Sahil Arora,Sourav Kalra,Anuhar Chaturvedi,Michael Heuser,Raj Kumar

Research Article

Diallyl Disulfide Inhibits Breast Cancer Stem Cell Progression and Glucose Metabolism by Targeting CD44/PKM2/AMPK Signaling

Journal: Current Cancer Drug Targets
Volume: 18 Issue: 6 Year: 2018 Page: 592-599
Author(s): Xinhua Xie,Xiaojia Huang,Hailin Tang,Feng Ye,Lu Yang,Xiaofang Guo,Zhi Tian,Xiaofang Xie,Cheng Peng,Xiaoming Xie

Research Article

Flavonoids as Pyruvate Kinase M2 Inhibitor: An In silico Analysis

Journal: Letters in Drug Design & Discovery
Volume: 21 Issue: 13 Year: 2024 Page: 2661-2673
Author(s):

Pyruvate Kinase M2: Regulatory Circuits and Potential for Therapeutic Intervention

Journal: Current Pharmaceutical Design
Volume: 20 Issue: 1 Year: 2014 Page: 2595-2606
Author(s): Vibhor Gupta, Kathryn E. Wellen, Sybille Mazurek, Rameshwar N. K. Bamezai

Fibroblast Growth Factor Receptor Inhibitors

Journal: Current Pharmaceutical Design
Volume: 19 Issue: 4 Year: 2013 Page: 687-701
Author(s): Suneel Kumar B.V.S, Lakshmi Narasu, Rambabu Gundla, Raveendra Dayam, Sarma J.A.R.P

Research Article

Integrated In Silico-In Vitro Discovery of Lung Cancer-related Tumor Pyruvate Kinase M2 (PKM2) Inhibitors

Journal: Medicinal Chemistry
Volume: 12 Issue: 7 Year: 2016 Page: 613-620
Author(s): Xiangyun Ye, Yinjia Sun, Yunhua Xu, Zhiwei Chen, Shun Lu

Research Article

Glycolysis Inhibitors for Anticancer Therapy: A Review of Recent Patents

Journal: Recent Patents on Anti-Cancer Drug Discovery
Volume: 11 Issue: 3 Year: 2016 Page: 297-308
Author(s): Huaming Sheng,Weijuan Tang

Review Article

Development of Pin1 Inhibitors and their Potential as Therapeutic Agents

Journal: Current Medicinal Chemistry
Volume: 27 Issue: 20 Year: 2020 Page: 3314-3329
Author(s): Yusuke Nakatsu,Yasuka Matsunaga,Koji Ueda,Takeshi Yamamotoya,Yuki Inoue,Masa-ki Inoue,Yu Mizuno,Akifumi Kushiyama,Hiraku Ono,Midori Fujishiro,Hisanaka Ito,Takayoshi Okabe,Tomoichiro Asano

Research Article

KIF20A Promotes CRC Progression and the Warburg Effect through theC-Myc/HIF-1α Axis

Journal: Protein & Peptide Letters
Volume: 31 Issue: 2 Year: 2024 Page: 107-115
Author(s):

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