Search Result "P-gp tracers"


Review Article

Importance of P-gp PET Imaging in Pharmacology

Journal: Current Pharmaceutical Design
Volume: 22 Issue: 38 Year: 2016 Page: 5830-5836
Author(s): Jun Toyohara

Carbon-11 Labeled Tracers for In Vivo Imaging of P-Glycoprotein Function: Kinetics, Advantages and Disadvantages

Journal: Current Topics in Medicinal Chemistry
Volume: 10 Issue: 1 Year: 2010 Page: 1820-1833
Author(s): Gert Luurtsema, Joost Verbeek, Mark Lubberink, Adriaan A. Lammertsma, Rudi Dierckx, Philip Elsinga, Albert D. Windhorst, Aren van Waarde

Review Article

Design and Synthesis of New Selective P-gp Substrates and Inhibitors

Journal: Current Pharmaceutical Design
Volume: 22 Issue: 38 Year: 2016 Page: 5774-5778
Author(s): Mariangela Cantore,Marcello Leopoldo,Francesco Berardi,Roberto Perrone,Nicola Antonio Colabufo

Three Decades of P-gp Inhibitors: Skimming Through Several Generations and Scaffolds

Journal: Current Medicinal Chemistry
Volume: 19 Issue: 13 Year: 2012 Page: 1946-2025
Author(s): A. Palmeira,E. Sousa,M. H. Vasconcelos,M. M. Pinto

Using PET Studies of P-gp Function to Elucidate Mechanisms Underlying the Disposition of Drugs

Journal: Current Topics in Medicinal Chemistry
Volume: 10 Issue: 1 Year: 2010 Page: 1799-1809
Author(s): Stina Syvanen, Margareta Hammarlund-Udenaes

11C-verapamil to Assess P-gp Function in Human Brain During Aging,Depression and Neurodegenerative Disease

Journal: Current Topics in Medicinal Chemistry
Volume: 10 Issue: 1 Year: 2010 Page: 1775-1784
Author(s): A. L. Bartels, O. L. de Klerk, R. Kortekaas, J. J. de Vries, K. L. Leenders

Modulation and Absorption of Xenobiotics: The Synergistic Role of CYP450 and P-gp Activities in Cancer and Neurodegenerative Disorders

Journal: Current Drug Metabolism
Volume: 12 Issue: 8 Year: 2011 Page: 702-712
Author(s): Carmela Inglese, Maria Grazia Perrone, Francesco Berardi, Roberto Perrone, Nicola Antonio Colabufo

Review Article

PET Tracers for Imaging of ABC Transporters at the Blood-Brain Barrier: Principles and Strategies

Journal: Current Pharmaceutical Design
Volume: 22 Issue: 38 Year: 2016 Page: 5779-5785
Author(s): Gert Luurtsema,Philip Elsinga,Rudi Dierckx,Ronald Boellaard,Aren van Waarde

Review Article

Kinetic Models for Measuring P-glycoprotein Function at the Blood-Brain Barrier with Positron Emission Tomography

Journal: Current Pharmaceutical Design
Volume: 22 Issue: 38 Year: 2016 Page: 5786-5792
Author(s): Mark Lubberink

Substrates, Inhibitors and Activators of P-glycoprotein: Candidates for Radiolabeling and Imaging Perspectives

Journal: Current Topics in Medicinal Chemistry
Volume: 10 Issue: 1 Year: 2010 Page: 1703-1714
Author(s): Nicola A. Colabufo, Francesco Berardi, Maria Grazia Perrone, Elena Capparelli, Mariangela Cantore, Carmela Inglese, Roberto Perrone

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