Search Result "Mechanism-based CYP inhibition"


Enzyme Kinetics for Clinically Relevant CYP Inhibition

Journal: Current Drug Metabolism
Volume: 6 Issue: 3 Year: 2005 Page: 241-257
Author(s): Zhi-Yi Zhang, Y. Nancy Wong

Potential Strategies for Minimizing Mechanism-Based Inhibition of Cytochrome P450 3A4

Journal: Current Pharmaceutical Design
Volume: 14 Issue: 1 Year: 2008 Page: 990-1000
Author(s): Shu-Feng Zhou

CYP Inhibition-Mediated Drug-Drug Interactions

Journal: Current Enzyme Inhibition
Volume: 6 Issue: 3 Year: 2010 Page: 130-145
Author(s): Karoly Tihanyi, Monika L. Bakk, Eva Hellinger, Monika Vastag

Letter Article

Mechanism-Based Inhibition of CYP3A Subfamilies by MacrolideAntibiotics and Piperine

Journal: Drug Metabolism and Bioanalysis Letters
Volume: 15 Issue: 2 Year: 2022 Page: 75-80
Author(s):

An In Vitro, High Throughput, Seven CYP Cocktail Inhibition Assay for the Evaluation of New Chemical Entities Using LC-MS/MS

Journal: Drug Metabolism Letters
Volume: 5 Issue: 1 Year: 2011 Page: 17-24
Author(s): Jennifer N. Otten, Gary P. Hingorani, Dylan P. Hartley, Scott D. Kragerud, Ronald B. Franklin

Mechanism-based Inhibition of CYP450: An Indicator of Drug-induced Hepatotoxicity

Journal: Current Drug Metabolism
Volume: 14 Issue: 9 Year: 2013 Page: 921-945
Author(s): Shan Feng,Xin He

Cytochrome P450 Enzymes Mechanism Based Inhibitors: Common Sub-Structures and Reactivity

Journal: Current Drug Metabolism
Volume: 6 Issue: 5 Year: 2005 Page: 413-451
Author(s): E. Fontana, P. M. Dansette, S. M. Poli

Therapeutic Drugs that Behave as Mechanism-Based Inhibitors of Cytochrome P450 3A4

Journal: Current Drug Metabolism
Volume: 5 Issue: 5 Year: 2004 Page: 415-442
Author(s): Shufeng Zhou, Eli Chan, Lee Yong Lim, Urs A. Boelsterli, Shu Chuen Li, Jiancheng Wang, Qiang Zhang, Min Huang, Anlong Xu

A Critical Evaluation of the Experimental Design of Studies of Mechanism Based Enzyme Inhibition, with Implications for In Vitro-In Vivo Extrapolation

Journal: Current Drug Metabolism
Volume: 7 Issue: 3 Year: 2006 Page: 315-334
Author(s): F. Ghanbari, K. Rowland-Yeo, J. C. Bloomer, S. E. Clarke, M. S. Lennard, G. T. Tucker, A. Rostami-Hodjegan

Role of Microtubules Network in CYP Genes Expression

Journal: Current Drug Metabolism
Volume: 6 Issue: 6 Year: 2005 Page: 545-552
Author(s): Z. Dvorak, J. Ulrichova, M. Modriansky

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