Search Result "Fragment based lead generation"


Fragment-Based Methods for Lead Discovery

Ebook: In Silico Lead Discovery
Volume: 1 Year: 2011
Author(s): Will R. Pitt,Alicia P. Higueruelo,Nikolay P. Todorov
Doi: 10.2174/978160805142711101010060

Fragment-based Designing for the Generation of Novel Leads Against BACE1

Journal: Central Nervous System Agents in Medicinal Chemistry
Volume: 15 Issue: 1 Year: 2015 Page: 52-64
Author(s): Sucharita Das,Sandipan Chakraborty,Soumalee Basu

From Fragment Screening to Potent Binders: Strategies for Fragment-to-Lead Evolution

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 9 Issue: 8 Year: 2009 Page: 956-961
Author(s): Krystian Eitner, Uwe Koch

New Lead Generation Strategies for Protein Kinase Inhibitors - Fragment Based Screening Approaches

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 4 Issue: 3 Year: 2004 Page: 301-311
Author(s): Adrian Gill

Fragment Library Screening and Lead Characterization Using SPR Biosensors

Journal: Current Topics in Medicinal Chemistry
Volume: 9 Issue: 1 Year: 2009 Page: 1725-1735
Author(s): U. Helena Danielson

Computational Techniques in Fragment Based Drug Discovery

Journal: Current Topics in Medicinal Chemistry
Volume: 7 Issue: 1 Year: 2007 Page: 1509-1513
Author(s): Hugo O. Villar, Mark R. Hansen

Library Design for Fragment Based Screening

Journal: Current Topics in Medicinal Chemistry
Volume: 5 Issue: 8 Year: 2005 Page: 751-762
Author(s): Ansgar Schuffenhauer, Simon Ruedisser, Andreas Marzinzik, Wolfgang Jahnke, Paul Selzer, Edgar Jacoby

An Integrated Approach to Fragment-Based Lead Generation:Philosophy, Strategy and Case Studies from AstraZenecas Drug Discovery Programmes

Journal: Current Topics in Medicinal Chemistry
Volume: 7 Issue: 1 Year: 2007 Page: 1600-1629
Author(s): Jeffrey S. Albert, Niklas Blomberg, Alexander L. Breeze, Alastair J. H. Brown, Jeremy N. Burrows, Philip D. Edwards, Rutger H. A. Folmer, Stefan Geschwindner, Ed J. Griffen, Peter W. Kenny, Thorsten Nowak, Lise-Lotte Olsson, Hitesh Sanganee, Adam B. Shapiro

Computational Tools for In Silico Fragment-Based Drug Design

Journal: Current Topics in Medicinal Chemistry
Volume: 12 Issue: 17 Year: 2012 Page: 1935-1943
Author(s): Jeremie Mortier,Christin Rakers,Raphael Frederick,Gerhard Wolber

Fragment Based Drug Design: From Experimental to Computational Approaches

Journal: Current Medicinal Chemistry
Volume: 19 Issue: 30 Year: 2012 Page: 5128-5147
Author(s): A. Kumar,A. Voet,K.Y.J. Zhang

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