Search Result "DNA-binding affinity and cytotoxicity"


Thiazole Containing Nitrogen Mustards: Synthesis, Structural Evaluation, Cytotoxicity and DNA Binding Studies

Journal: Letters in Drug Design & Discovery
Volume: 8 Issue: 9 Year: 2011 Page: 838-842
Author(s): Nulgulmnalli Manjunathiah Raghavendra, Surampudi Renuka, Sayan Dutta Gupta, Pingili Divya

Determination of Binding Constant of DNA-binding Drug to Target DNA by Surface Plasmon Resonance Biosensor Technology

Journal: Current Drug Targets - Immune, Endocrine & Metabolic Disorders
Volume: 5 Issue: 1 Year: 2005 Page: 61-72
Author(s): Liang-Ping Lin, Long-Sun Huang, Chii-Wann Lin, Chi-Kung Lee, Ji-Liang Chen, Su-Ming Hsu, Shiming Lin

Anticancer Activity and DNA Binding of 4-Alkylenediamines Modified Naphthalimide Derivatives

Journal: Letters in Drug Design & Discovery
Volume: 11 Issue: 6 Year: 2014 Page: 742-748
Author(s): Ke-Rang Wang,Feng Qian,Zi-Bo Yang,Hong-Wei An,Dan Han,Hua Chen,Ping-Zhu Zhang,Xiao-Liu Li

The DNA-Binding and Bioactivity of Rare Earth Metal Complexes

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 13 Issue: 1 Year: 2013 Page: 1487-1500
Author(s): Li Yang, Bochu Wang, Jun Tan, Liancai Zhu

Amplification of Anticancer Drug-Induced DNA Damage and Apoptosis by DNA-Binding Compounds

Journal: Current Medicinal Chemistry - Anti-Cancer Agents
Volume: 4 Issue: 5 Year: 2004 Page: 415-419
Author(s): Shosuke Kawanishi, Yusuke Hiraku

Is DNA Minor Groove Binding Crucial for Biological Activity of Triazoloacridinones with Cytotoxic and Antitumour Properties?

Journal: Letters in Drug Design & Discovery
Volume: 6 Issue: 4 Year: 2009 Page: 242-245
Author(s): Marcin Koba, Katarzyna Koba, Tomasz Baczek

Synthesis of Benzopyran Linked Pyrrolo[2,1-c][1,4]benzodiazepines as DNA-Binding and Potential Anticancer Agents

Journal: Medicinal Chemistry
Volume: 9 Issue: 2 Year: 2013 Page: 177-192
Author(s): Ahmed Kamal,Rajender,Methuku Kashi Reddy,Vangala Santhosh Reddy,Gajjela Bharath Kumar

Therapeutic Agents Based on DNA Sequence Specific Binding

Journal: Current Topics in Medicinal Chemistry
Volume: 15 Issue: 14 Year: 2015 Page: 1293-1322
Author(s): Luke Pett,John A. Hartley,Konstantinos Kiakos

Synthesis, DNA Binding Ability and Anticancer Activity of 2-heteroaryl Substituted Benzimidazoles Linked Pyrrolo[2,1-c][1,4]benzodiazepine Conjugates

Journal: Medicinal Chemistry
Volume: 9 Issue: 5 Year: 2013 Page: 651-659
Author(s): Ahmed Kamal,Praveen Kumar Pogula,Mohammed Naseer Ahmed Khan,Bobburi Naga Seshadri,Kokkonda Sreekanth

Chemometric Evaluation of the Significance of Molecular Structural Descriptors on Binding of Acridinone Derivatives to DNA

Journal: Letters in Drug Design & Discovery
Volume: 7 Issue: 7 Year: 2010 Page: 494-499
Author(s): Marcin Koba, Tomasz Baczek

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