Search Result "Bridged piperazine"


Bridged Piperazines and Piperidines as CCR1 Antagonists with Oral Activity in Models of Arthritis and Multiple Sclerosis

Journal: Letters in Drug Design & Discovery
Volume: 3 Issue: 1 Year: 2006 Page: 689-694
Author(s): Laszlo Revesz, Birgit Bollbuck, Thomas Buhl, Janet Dawson, Roland Feifel, Richard Heng, Peter Hiestand, Helmut Sparrer, Achim Schlapbach, Rudolf Waelchli, Pius Loetscher

Mini-Review Article

Synthetic Protocols, Structural Activity Relationship, and BiologicalActivity of Piperazine and its Derivatives

Journal: Medicinal Chemistry
Volume: 20 Issue: 8 Year: 2024 Page: 753-780
Author(s):

Stereoselective Synthesis of Polysubstituted Piperazines and Oxopiperazines. Useful Building Blocks in Medicinal Chemistry

Journal: Current Topics in Medicinal Chemistry
Volume: 14 Issue: 10 Year: 2014 Page: 1308-1316
Author(s): Alessandro Mordini,Gianna Reginato,Massimo Calamante,Lorenzo Zani

General Research Article

Novel Tri-substituted Thiazoles Bearing Piperazine Ring: Synthesis and Evaluation of their Anticancer Activity

Journal: Letters in Drug Design & Discovery
Volume: 16 Issue: 5 Year: 2019 Page: 547-555
Author(s): Asaf Evrim Evren,Leyla Yurttaş,Busra Eksellı,Gulsen Akalın-Cıftcı

Research Article

Novel Piperazine Amides of Cinnamic Acid Derivatives as Tyrosinase Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 16 Issue: 1 Year: 2019 Page: 36-44
Author(s): Zehra Tuğçe Gür,Fatma Sezer Şenol,Suhaib Shekfeh,İlkay Erdoğan Orhan,Erden Banoğlu,Burcu Çalişkan

Synthetic Chemistry with N-Acyliminium Ions Derived from Piperazine-2,5-Diones and Related Compounds

Journal: Current Organic Synthesis
Volume: 6 Issue: 2 Year: 2009 Page: 143-168
Author(s): Carmen Avendano, Elena de la Cuesta

Synthesis of Thiophenyl Schiff Bases via Buchwald-Hartwig Coupling of Piperazines to Quinoline Motif

Journal: Current Organic Synthesis
Volume: 11 Issue: 4 Year: 2014 Page: 621-625
Author(s): Rahul V. Patel,Se Won Park

N,N-Bis(trifluoromethylquinolin-4-yl)diamino Alkanes: Synthesis and Antimalarial Activity

Journal: Medicinal Chemistry
Volume: 4 Issue: 5 Year: 2008 Page: 438-445
Author(s): Joseph L. Kgokong, Gilbert M. Matsabisa, Peter P. Smith, Jaco C. Breytenbach

Research Article

Synthesis, Antimicrobial, Antioxidant and Molecular Docking Studies on Novel 6-Methoxybenzothiazole-piperazine Derivatives with Propanamide Chain

Journal: Current Topics in Medicinal Chemistry
Volume: 20 Issue: 19 Year: 2020 Page: 1733-1741
Author(s): Nesrin Atiah Alhusadi,Bengisu Turgutalp,Inci Deniz,Ebru Turkoz Acar,Hande Sipahi,Mine Yarim,Enise Ece Gurdal

Discovery of Novel Lead in the Group of N-substituted Piperazine Ether Derivatives with Potential Histamine H3 Receptor Activity

Journal: Medicinal Chemistry
Volume: 10 Issue: 6 Year: 2014 Page: 588-599
Author(s): Kamil J. Kuder, Marta Stachnik, Walter Schunack, Ewa Szyman ska, Katarzyna Kiec -Kononowicz

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