Search Result "BET inhibitors"
BET Inhibitors as Anticancer Agents: A Patent Review
Journal: Recent Patents on Anti-Cancer Drug Discovery
Volume: 12 Issue: 4 Year: 2017 Page: 340-364
Author(s): Imran Ali,Gildon Choi,Kwangho Lee
Small-Molecule BET Inhibitors in Clinical and Preclinical Development and Their Therapeutic Potential
Journal: Current Topics in Medicinal Chemistry
Volume: 15 Issue: 8 Year: 2015 Page: 776-794
Author(s): Lei Yu,Zhen Wang,Zhang Zhang,Xiaomei Ren,Xiaoyun Lu,Ke Ding
Disrupting Acetyl-lysine Interactions: Recent Advance in the Development of BET Inhibitors
Journal: Current Drug Targets
Volume: 19 Issue: 10 Year: 2018 Page: 1148-1165
Author(s): Fa Zhang,Shutao Ma
The BET-Bromodomain Inhibitor JQ1 Reduces Inflammation and Tau Phosphorylation at Ser396 in the Brain of the 3xTg Model of Alzheimerâs Disease
Journal: Current Alzheimer Research
Volume: 13 Issue: 9 Year: 2016 Page: 985-995
Author(s): Marco Magistri,Dmitry Velmeshev,Madina Makhmutova,Prutha Patel,Gregory C. Sartor,Claude-Henry Volmar,Claes Wahlestedt,Mohammad Ali Faghihi
Recent Developments in Targeting Bromodomain and Extra TerminalDomain Proteins for Cancer Therapeutics
Journal: Current Medicinal Chemistry
Volume: 29 Issue: 25 Year: 2022 Page: 4391-4409
Author(s):
The Bromodomain and Extra-Terminal Protein Inhibitor OTX015 Suppresses T Helper Cell Proliferation and Differentiation
Journal: Current Molecular Medicine
Volume: 18 Issue: 9 Year: 2018 Page: 594-601
Author(s): Xiao Hu,Lauren P. Schewitz-Bowers,Philippa J. P. Lait,David A. Copland,Madeleine L. Stimpson,Jing Jing Li,Yizhi Liu,Andrew D. Dick,Richard W. J. Lee,Lai Wei
Prediction of Inhibition Activity of BET Bromodomain Inhibitors using Grid Search-Based Extreme Learning Machine and Molecular Docking
Journal: Letters in Drug Design & Discovery
Volume: 18 Issue: 11 Year: 2021 Page: 1039-1049
Author(s): Oluwatoba Emmanuel Oyeneyin,Babatunde Samuel Obadawo,Segun Michael Orimoloye,Eric Oluwafisayo Akintemi,Nureni Ipinloju,Adeola M. Asere,Taoreed O. Owolabi
Overexpression of Bromodomain and Extraterminal Domain is Associated withProgression, Metastasis and Unfavorable Outcomes: Highlighting Prognostic andTherapeutic Value of the BET Protein Family in Gastric Cancer
Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 23 Issue: 7 Year: 2023 Page: 794-806
Author(s): Shahrzad S. Fard,Seyed A. Mousavi,Seyed H. Ghaffari
Charting the Bromodomain BRD4: Towards the Identification of Novel Inhibitors with Molecular Similarity and Receptor Mapping
Journal: Letters in Drug Design & Discovery
Volume: 15 Issue: 9 Year: 2018 Page: 1002-1011
Author(s): Fernando D. Prieto-Martinez,Jose L. Medina-Franco
JQ1, a BET Inhibitor, Synergizes with Cisplatin and Induces Apoptosis in Highly Chemoresistant Malignant Pleural Mesothelioma Cells
Journal: Current Cancer Drug Targets
Volume: 18 Issue: 8 Year: 2018 Page: 816-828
Author(s): Ilaria Zanellato,Donato Colangelo,Domenico Osella