Search Result "Agonists vs. antagonists binding"


Medicinal Chemistry of P2X Receptors: Agonists and Orthosteric Antagonists

Journal: Current Medicinal Chemistry
Volume: 22 Issue: 7 Year: 2015 Page: 915-928
Author(s): Catia Lambertucci,Diego Dal Ben,Michela Buccioni,Gabriella Marucci,Ajiroghene Thomas,Rosaria Volpini

A2A Adenosine Receptor and its Modulators: Overview on a Druggable GPCR and on Structure-Activity Relationship Analysis and Binding Requirements of Agonists and Antagonists

Journal: Current Pharmaceutical Design
Volume: 14 Issue: 1 Year: 2008 Page: 1525-1552
Author(s): G. Cristalli, C. Lambertucci, G. Marucci, R. Volpini, D. Dal Ben

Glutamate Receptor Agonists: Stereochemical Aspects

Journal: Current Topics in Medicinal Chemistry
Volume: 11 Issue: 7 Year: 2011 Page: 887-906
Author(s): Stine Byskov Vogensen, Jeremy R. Greenwood, Lennart Bunch, Rasmus Praetorius Clausen

GnRH Agonists and Antagonists in Cancer Therapy

Journal: Current Medicinal Chemistry - Anti-Cancer Agents
Volume: 3 Issue: 6 Year: 2003 Page: 399-410
Author(s): Murty V. Chengalvala, Jeffrey C. Pelletier, Gregory S. Kopf

Recent Advances in Identification and Characterization of β-Adrenoceptor Agonists and Antagonists

Journal: Current Topics in Medicinal Chemistry
Volume: 7 Issue: 2 Year: 2007 Page: 207-216
Author(s): J. Paul Hieble

Selective Agonists and Antagonists for Kainate Receptors

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 2 Issue: 2 Year: 2002 Page: 177-184
Author(s): Paola Conti, Marco De Amici, Carlo De Micheli

Receptor-Binding and Pharmacokinetic Properties of Dopaminergic Agonists

Journal: Current Topics in Medicinal Chemistry
Volume: 8 Issue: 1 Year: 2008 Page: 1049-1067
Author(s): Trond Kvernmo, John Houben, Ingebrigt Sylte

The Evolution of Histamine H3 Antagonists/Inverse Agonists

Journal: Current Topics in Medicinal Chemistry
Volume: 11 Issue: 6 Year: 2011 Page: 648-660
Author(s): Evan P. Lebois, Carrie K. Jones, Craig W. Lindsley

Strategies for Design of Non Peptide CCK1R Agonist/Antagonist Ligands

Journal: Current Topics in Medicinal Chemistry
Volume: 7 Issue: 1 Year: 2007 Page: 1180-1194
Author(s): M. Teresa Garcia-Lopez, Rosario Gonzalez-Muniz, Mercedes Martin-Martinez, Rosario Herranz

Development of Selective High Affinity Antagonists, Agonists, and Radioligands for the P2Y1 Receptor

Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 11 Issue: 6 Year: 2008 Page: 410-419
Author(s): Dayle Houston, Stefano Costanzi, Kenneth A. Jacobson, T. Kendall Harden

Previous   Next

Go To   Results 1 - 1 of 2333

Apply Filters

Volume Years
Article Type
Publication Title
Subject Title

Content Type


Ads
© 2024 Bentham Science Publishers | Privacy Policy