Search Result "20-dione"


General Research Article

The Synthesis, Anticancer Activity, Structure-Activity Relationships and Molecular Modelling Studies of Novel Isoindole-1,3(2H)-dione Compounds Containing Different Functional Groups

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 20 Issue: 11 Year: 2020 Page: 1368-1378
Author(s): Ayse Tan,Serap Kizilkaya,Unzile Kelestemur,Atilla Akdemir,Yunus Kara

Non-Selective Inhibition of Cyclooxygenase Enzymes by Aminoacetylenic Isoindoline 1,3-Diones

Journal: Inflammation & Allergy - Drug Targets (Discontinued)
Volume: 11 Issue: 5 Year: 2012 Page: 369-374
Author(s): Nidal A. Qinna,Zuhair A. Muhi-eldeen,Mohammad Ghattas,Tawfiq M. Alhussainy,Jenan Al-Qaisi,Khalid Z. Matalka

Research Article

Mandelic Acid: An Efficient Organo-catalyst for the Synthesis of 3-substituted-3- Hydroxy-indolin-2-ones and Related Derivatives in Aqueous Ethanol at Room Temperature

Journal: Current Organocatalysis
Volume: 8 Issue: 1 Year: 2021 Page: 147-159
Author(s): Gurpreet Kaur,Rajat Kumar,Shivam Saroch,Vivek Kumar Gupta,Bubun Banerjee

Guggulsterone for Chemoprevention of Cancer

Journal: Current Pharmaceutical Design
Volume: 22 Issue: 3 Year: 2016 Page: 294-306
Author(s): Shishir Shishodia,Nkem Azu,Jason A. Rosenzweig,Desiree A. Jackson

Aldose Reductase Inhibitory Potential of Several Thiazolyl-thiazolidine- 2,4-Diones

Journal: Letters in Drug Design & Discovery
Volume: 10 Issue: 5 Year: 2013 Page: 415-419
Author(s): Net Das-Evcimen, Mutlu Sar?kaya, A. Selen Gurkan-Alp, Oya Bozdag-Dundar

Research Article

A Novel Scheme for the Synthesis of 21-Acetoxypregna-1,4,9(11)-triene- 17α,21-diol-3,20-dione from 9α-Hydroxyandrostenedione

Journal: Current Bioactive Compounds
Volume: 16 Issue: 5 Year: 2020 Page: 606-610
Author(s): Nguyen T. Diep,Luu D. Huy

Research Article

UHPLC Quantitation Method for New Thiazolidinedione LPSF/GQ-02 and In Vitro/In Vivo Kinetic Studies

Journal: Drug Metabolism Letters
Volume: 10 Issue: 3 Year: 2016 Page: 206-212
Author(s): Carla Monalizi Vieira,Michel Leandro de Campos,Elias Carvalho Padilha,Marina Pitta,Ivan da Rocha Pitta,Maria do Carmo Alves de Lima,Rosângela Gonçalves Peccinini

Research Article

An Efficient Procedure for the Synthesis of 21-Acetoxypregna-1,4,9(11),16- tetraene-3,20-dione

Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 23 Issue: 3 Year: 2020 Page: 225-231
Author(s): Luu D. Huy,Nguyen T. Diep,Tran K. Vu,Tatiana S. Savinova,Marina V. Donova

Virtual Screening and Discovery of Novel Aurora Kinase Inhibitors

Journal: Current Topics in Medicinal Chemistry
Volume: 14 Issue: 17 Year: 2014 Page: 2006-2019
Author(s): R. Raghu,Vinod Devaraji,K. Leena,Sd. Riyaz,Polavaru Baby Rani,Suneel Kumar. B,Pradeep Kumar Naik,P.K. Dubey,Devadasan Velmurugan,M. Vijayalakshmi

Mitoxantrone Targets the ATP-binding Site of FAK, Binds the FAK Kinase Domain and Decreases FAK, Pyk-2, c-Src, and IGF-1R In Vitro Kinase Activities

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 13 Issue: 4 Year: 2013 Page: 546-554
Author(s): Vita M. Golubovskaya, Baotran Ho, Min Zheng, Andrew Magis, David Ostrov, William G. Cance

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