Search Result "selective JAK1."


General Research Article

Design and Synthesis of New JAK1 Inhibitors based on Sulfonamide-Triazine Conjugates

Journal: Current Computer-Aided Drug Design
Volume: 17 Issue: 7 Year: 2021 Page: 916-926
Author(s): Safa Daoud,Mutasem O. Taha

Clinical Confirmation that the Selective JAK1 Inhibitor Filgotinib (GLPG0634) has a Low Liability for Drug-drug Interactions

Journal: Drug Metabolism Letters
Volume: 10 Issue: 1 Year: 2016 Page: 38-48
Author(s): Florence Namour,Julie Desrivot,Annegret Van der Aa,Pille Harrison,Gerben van`t Klooster,Chantal Tasset

Perspective

Abrocitinib: First Globally Approved Selective Janus Kinase-1 Inhibitorfor the Treatment of Atopic Dermatitis

Journal: Current Medicinal Chemistry
Volume: 30 Issue: 38 Year: 2023 Page: 4278-4282
Author(s): Surya K. De

Review Article

Searching for Novel Janus Kinase-2 Inhibitors Using a Combination of Pharmacophore Modeling, 3D-QSAR Studies and Virtual Screening

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 17 Issue: 3 Year: 2017 Page: 268-294
Author(s): Eleni Vrontaki,Georgia Melagraki,Antreas Afantitis,Thomas Mavromoustakos,George Kollias

Perspective

First Approval of Pacritinib as a Selective Janus Associated Kinase-2 Inhibitor forthe Treatment of Patients with Myelofibrosis

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 23 Issue: 12 Year: 2023 Page: 1355-1360
Author(s): Surya K. De

Review Article

Current Status in the Discovery of Covalent Janus Kinase 3 (JAK3) Inhibitors

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 19 Issue: 18 Year: 2019 Page: 1531-1543
Author(s): Jun Dai,LiXi Yang,Glynn Addison

Insights into the Structural Features Essential for JAK2 Inhibition and Selectivity

Journal: Current Medicinal Chemistry
Volume: 23 Issue: 13 Year: 2016 Page: 1331-1355
Author(s): Chao Zhao,Daulat Bikram Khadka,Won-Jea Cho

Mini-Review Article

Approach in Improving Potency and Selectivity of Kinase Inhibitors: Allosteric Kinase Inhibitors

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 21 Issue: 8 Year: 2021 Page: 991-1003
Author(s): Shangfei Wei,Tianming Zhao,Jie Wang,Xin Zhai

Review Article

An Update on JAK Inhibitors

Journal: Current Medicinal Chemistry
Volume: 26 Issue: 10 Year: 2019 Page: 1806-1832
Author(s): Francesca Musumeci,Chiara Greco,Ilaria Giacchello,Anna Lucia Fallacara,Munjed M. Ibrahim,Giancarlo Grossi,Chiara Brullo,Silvia Schenone

Chemical Genomic and Proteomic Methods for Determining Kinase Inhibitor Selectivity

Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 10 Issue: 8 Year: 2007 Page: 652-666
Author(s): Ratika Krishnamurty, Dustin J. Maly

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