Search Result "receptor kinetics"


Kinetic and Structural Determinants for GABA-A Receptor Potentiation by Neuroactive Steroids

Journal: Current Neuropharmacology
Volume: 8 Issue: 1 Year: 2010 Page: 18-25
Author(s): Gustav Akk, Douglas F. Covey, Alex S. Evers, Steven Mennerick, Charles F. Zorumski, Joe Henry Steinbach

The Role of Binding Kinetics in GPCR Drug Discovery

Journal: Current Topics in Medicinal Chemistry
Volume: 15 Issue: 24 Year: 2015 Page: 2504-2522
Author(s): David C. Swinney,Brad A. Haubrich,Isabelle Van Liefde,Georges Vauquelin

Kinetic Analysis of the Cleavage of Human Protease-Activated Receptor-1 / 2 / 3 and 4 Using Quenched-Fluorescent Peptide Substrates

Journal: Protein & Peptide Letters
Volume: 9 Issue: 5 Year: 2002 Page: 387-393
Author(s): Mark T. Fox, Brett Greer, Jill Lawson, Adrienne Healy, Patrick Harriott

Novel Experimental Design for Steady-state Processes: A Systematic Bayesian Approach for Enzymes, Drug Transport, Receptor Binding, Continuous Culture and Cell Transport Kinetics

Journal: Medicinal Chemistry
Volume: 1 Issue: 1 Year: 2005 Page: 21-29
Author(s): M. James C. Crabbe, Emma F. Murphy, Steven G. Gilmour

Review Article

Non-peptide CRF-Receptor Antagonists: Allosterism, Kinetics and Translation to Efficacy in Human Disease

Journal: Current Molecular Pharmacology
Volume: 10 Issue: 4 Year: 2017 Page: 282-295
Author(s): Samuel R.J. Hoare,Dimitri E. Grigoriadis

Review Article

Kinetic Resolutions Enabled by N-Heterocyclic Carbene Catalysis

Journal: Current Organic Synthesis
Volume: 14 Issue: 5 Year: 2017 Page: 654-664
Author(s): Shuang Yang, Xinqiang Fang

The Role of Kinetics in High Throughput Screening for Drugs

Ebook: Young People’s Visions of the World
Volume: 1 Year: 2010
Author(s): Agustina Gomez-Hens, M Paz Aguilar-Caballos
Doi: 10.2174/97816080519911050101

Kinetics of Vascular Targeted Monoclonal Antibody

Journal: Current Drug Delivery
Volume: 7 Issue: 5 Year: 2010 Page: 428-435
Author(s): Stephen J. Kennel, Ying Huang, Wen- Bin Zeng, Alan Stuckey, Jonathan Wall

Review Article

Roles of Accelerated Molecular Dynamics Simulations in Predictions ofBinding Kinetic Parameters

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 24 Issue: 14 Year: 2024 Page: 1323-1333
Author(s):

Drug Design for Protein Kinases and Phosphatases: Flexible-Receptor Docking, Binding Affinity and Specificity, and Drug-Binding Kinetics

Journal: Current Pharmaceutical Design
Volume: 19 Issue: 26 Year: 2013 Page: 4739-4754
Author(s): Chung F. Wong,Sneha Bairy

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