Search Result "pyrimidine-2(1H)-thiones"


Highly Efficient, Chemoselective Syntheses of 2-Methoxy-4-substituted Pyrimidines

Journal: Letters in Organic Chemistry
Volume: 8 Issue: 8 Year: 2011 Page: 545-548
Author(s): Chunyan Xu, Chuanjie Cheng, Hongtao Liu, Bo Liu

Letter Article

Synthesis of Substituted imidazo [1, 5-a] pyrimidine-2-(1H)-one Core Structure

Journal: Current Organic Synthesis
Volume: 17 Issue: 1 Year: 2020 Page: 23-28
Author(s): Vijay Kalhapure,Dhananjay Magar,Nishant Kothalkar,Tushar Khaladkar,Abhijit Roychowdhury

Synthesis of 4-(5-chloro-3-methyl-1-phenyl-1H-pyrazol-4-yl)-6-(substituted phenyl)pyrimidin-2-ol Analogues as Anti-Inflammatory and Analgesic Agents

Journal: Letters in Drug Design & Discovery
Volume: 10 Issue: 8 Year: 2013 Page: 776-782
Author(s): Muhammad Jahangir Alam,Mohamed Jawed Ahsan,Ozair Alam,Suroor Ahmad Khan

Research Article

Discovery of N-Phenyl-4-(1H-pyrrol-3-yl)pyrimidin-2-amine Derivatives as Potent Mnk2 Inhibitors: Design, Synthesis, SAR Analysis, and Evaluation of in vitro Anti-leukaemic Activity

Journal: Medicinal Chemistry
Volume: 15 Issue: 6 Year: 2019 Page: 602-623
Author(s): Ahmed M. Abdelaziz,Sarah Diab,Saiful Islam,Sunita K.C. Basnet,Benjamin Noll,Peng Li,Laychiluh B. Mekonnen,Jingfeng Lu,Hugo Albrecht,Robert W. Milne,Cobus Gerber,Mingfeng Yu,Shudong Wang

Novel 2-hydrazino-pyrimidin-4(3H)-one Derivatives with Pseudofunctional- Similarity to Siderophores as Potential Antimycobacterial Agents

Journal: Medicinal Chemistry
Volume: 9 Issue: 1 Year: 2013 Page: 77-83
Author(s): Ranjeet Bairwa, Nilesh R. Tawari, Amruta Alate, Swapnil Anam, Mariam S. Degani, Muktikant Ray, Ramakrishna M. G. Rajan

Research Article

Synthesis, Cytotoxicity, ADMET and Molecular Docking Studies of Some Quinoline-Pyrimidine Hybrid Compounds: 3-(2-Amino-6-arylpyrimidin-4- yl)-4-hydroxy-1-methylquinolin-2(1H)-ones

Journal: Medicinal Chemistry
Volume: 18 Issue: 1 Year: 2022 Page: 36-50
Author(s): Duong Ngoc Toan,Nguyen Dinh Thanh,Mai Xuan Truong,Dinh Thuy Van

Research Article

Synthesis of Some Novel 5,7-Disubstituted-2-phenyl-5H-[1,3,4]thiadiazolo [3,2-a]pyrimidine Derivatives and Evaluation of Their Biological Activity

Journal: Letters in Organic Chemistry
Volume: 13 Issue: 9 Year: 2016 Page: 661-671
Author(s): Talavara Venkatesh,Yadav D. Bodke,Nibin M. Joy,B. M. Vinoda,Yallappa Shiralgi,B. L. Dhananjaya

4-Thiophenoxy-N-(3,4,5-Trialkoxyphenyl)Pyrimidine-2-Amines as Potent and Selective Inhibitors of the T-Cell Tyrosine Kinase p56lck

Journal: Current Medicinal Chemistry
Volume: 11 Issue: 6 Year: 2004 Page: 747-753
Author(s): D. F.C. Moffat, R. A. Allen, S. E. Rapecki, P. D. Davis, J. OConnell, M. C. Hutchings, M. A. King, B. A. Boyce, M. J. Perry

Research Article

Antihelminthic Activity of Some 2-Substituted Thieno[2,3-d]pyrimidin-4-ones

Journal: Letters in Drug Design & Discovery
Volume: 15 Issue: 8 Year: 2018 Page: 887-894
Author(s): Anelia Mavrova,Stefan Dimov,Dimitar Vuchev,Kameliya Anichina,Denitsa Yancheva

Journal: Letters in Organic Chemistry
Volume: 8 Issue: 6 Year: 2011 Page: 401-405
Author(s): Mohammad Bakherad, Ali Keivanloo, Marzieh Mohammadi, Saeideh Jajarmi

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