Search Result "pyrazolopyrimidines"


General Review Article

Medicinal Chemistry of Pyrazolopyrimidine Scaffolds Substituted with DifferentHeterocyclic Nuclei

Journal: Current Pharmaceutical Design
Volume: 28 Issue: 41 Year: 2022 Page: 3374-3403
Author(s): Galal H. elgemeie,Rasha A. Azzam,Wafaa A. Zaghary,Mohammed A. Khedr,Gihad E. Elsherif

Research Article

Synthesis of β-Amino Carbonyl 6-(Aminomethyl)- and6-(Hydroxymethyl)pyrazolopyrimidines for DPP-4 Inhibition Study

Journal: Current Medicinal Chemistry
Volume: 31 Issue: 22 Year: 2024 Page: 3380-3396
Author(s): Henry J. Tsai,Fung Fuh Wong

Research Article

Novel 1,3,4-trisubstituted Pyrazolopyrimidine Derivatives Show PotentAntiproliferative Activity in Mantle Cell Lymphoma

Journal: Letters in Drug Design & Discovery
Volume: 21 Issue: 11 Year: 2024 Page: 2063-2071
Author(s):

Evaluation of Novel 7-(hetero)aryl-substituted Pyrazolo[1, 5-a]pyrimidines as Phosphodiesterase-4 Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 7 Issue: 6 Year: 2010 Page: 402-408
Author(s): Arumugam Kodimuthali, Rajesh Gupta, Kishore Venkata Laxmi Parsa, Padala Lakshmi Prasunamba, Manojit Pal

GABAA Receptor Specific Pyrazolopyrimidines as Potential Imaging Agents: In Vivo Characteristics of a New 18F-labelled Indiplon Derivative

Journal: Current Radiopharmaceuticals
Volume: 2 Issue: 1 Year: 2009 Page: 24-31
Author(s): W. Deuther-Conrad, S. Fischer, M. Scheunemann, A. Hiller, M. Diekers, A. Friemel, F. Wegner, J. Steinbach, A. Hoepping, P. Brust

Pyrazolopyrimidine Derivatives as Antineoplastic Agents: with a Special Focus on Thyroid Cancer

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 16 Issue: 2 Year: 2016 Page: 86-93
Author(s): Silvia Martina Ferrari,Concettina La Motta,Stefania Sartini,Enke Baldini,Gabriele Materazzi,Ugo Politti,Ilaria Ruffilli,Salvatore Ulisse,Paolo Miccoli,Alessandro Antonelli,Poupak Fallahi

Studies on the Chemical Reactivity of Ethyl 4-sulfanyl-6-methyl-2-phenylpyrimidine-5-carboxylate

Journal: Current Organic Chemistry
Volume: 15 Issue: 1 Year: 2011 Page: 1661-1668
Author(s): A. H. Moustafa, M. G. Assy, A. E. Amr, R. M. Saber

Microwave Synthesis of Guanine and Purine Analogs

Journal: Current Microwave Chemistry
Volume: 1 Issue: 2 Year: 2014 Page: 155-176
Author(s): Galal Elgemeie,Mai Hamed

Research Article

Pyrrolopyrazoles: Synthesis, Evaluation and Pharmacological Screening as Antidepressant Agents

Journal: Medicinal Chemistry
Volume: 15 Issue: 8 Year: 2019 Page: 911-922
Author(s): Samar S. Fatahala,Shahira Nofal,Eman Mahmoud,Rania H. Abd El-hameed

Research Article

New Route to the Synthesis of Novel Pyrazolo[1,5-a]pyrimidines andEvaluation of their Antimicrobial Activity as RNA Polymerase Inhibitors

Journal: Medicinal Chemistry
Volume: 18 Issue: 9 Year: 2022 Page: 926-948
Author(s): Amira E. M. Abdallah,Galal H. Elgemeie

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