Search Result "inverse agonism"


Intrinsic Activity at Adenosine A1 Receptors: Partial and Inverse Agonism

Journal: Current Pharmaceutical Design
Volume: 8 Issue: 2 Year: 2002 Page: 2333-2344
Author(s): Rianne A.F. de Ligt, Ad P. Ijzerman

Atypical antipsychotics and inverse agonism at 5-HT2 receptors

Journal: Current Pharmaceutical Design
Volume: 21 Issue: 26 Year: 2015 Page: 3732-3738
Author(s): Laura C. Sullivan,William P Clarke,Kelly A. Berg

Cannabinoid Receptor G Protein-Coupling and Inverse Agonism

Journal: Current Neuropharmacology
Volume: 2 Issue: 1 Year: 2004 Page: 31-36
Author(s): Deborah L. Lewis

A Pharmacological Primer of Biased Agonism

Journal: Endocrine, Metabolic & Immune Disorders - Drug Targets
Volume: 11 Issue: 2 Year: 2011 Page: 92-98
Author(s): Bradley T. Andresen

Drugs that Act Through Membrane Receptors and Involve an Action of Inverse Agonism

Ebook: Frontiers in CNS Drug Discovery
Volume: 1 Year: 2010
Author(s): Gabriel Barreda-Gomez, Rafael Rodriguez-Puertas
Doi: 10.2174/978160805159511001010413

Development of New Drugs that Act Through Membrane Receptors and Involve an Action of Inverse Agonism

Journal: Recent Patents on CNS Drug Discovery (Discontinued)
Volume: 1 Issue: 2 Year: 2006 Page: 207-217
Author(s): Rafael Rodriguez-Puertas, Gabriel Barreda-Gomez

Review Article

δ Opioid Receptor Inverse Agonists and their In Vivo Pharmacological Effects

Journal: Current Topics in Medicinal Chemistry
Volume: 20 Issue: 31 Year: 2020 Page: 2889-2902
Author(s): Shigeto Hirayama,Hideaki Fujii

Assessing Receptor Affinity for Inverse Agonists: Schild and Cheng-Prusoff Methods Revisited

Journal: Current Drug Targets
Volume: 8 Issue: 1 Year: 2007 Page: 197-202
Author(s): Jesus Giraldo, Juan Serra, David Roche, Xavier Rovira

Angiotensin II Receptor Blocker as an Inverse Agonist: A Current Perspective

Journal: Current Hypertension Reviews
Volume: 1 Issue: 2 Year: 2005 Page: 115-121
Author(s): Shin-ichiro Miura, Masahiro Fujino, Keijiro Saku

Biased Agonism at the Parathyroid Hormone Receptor: A Demonstration of Functional Selectivity in Bone Metabolism

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 12 Issue: 9 Year: 2012 Page: 856-865
Author(s): B. N. Bohinc,D. Gesty-Palmer

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