Search Result "dualsteric ligand"


Review Article

Dopamine D2 Receptors Dimers: How can we Pharmacologically Target Them?

Journal: Current Neuropharmacology
Volume: 16 Issue: 2 Year: 2018 Page: 222-230
Author(s): Marco Carli,Shivakumar Kolachalam,Stefano Aringhieri,Mario Rossi,Luca Giovannini,Roberto Maggio,Marco Scarselli

Review Article

Recent Advances in the Drug Discovery and Development of Dualsteric/ Bitopic Activators of G Protein-Coupled Receptors

Journal: Current Topics in Medicinal Chemistry
Volume: 19 Issue: 2 Year: 2019 Page: 2378-2392
Author(s): Bethany A. Reinecke,Huiqun Wang,Yan Zhang

A Hydrazide Linker Strategy for Heterobivalent Compounds as Ortho- and Allosteric Ligands of Acetylcholine-Binding Proteins

Journal: Current Topics in Medicinal Chemistry
Volume: 11 Issue: 2 Year: 2011 Page: 2731-2748
Author(s): Paul W. Elsinghorst, Wolfgang Hartig, Daniela Gundisch, Klaus Mohr, Christian Trankle, Michael Gutschow

Review Article

Analgesic Effects Mediated by Muscarinic Receptors: Mechanisms and Pharmacological Approaches

Journal: Central Nervous System Agents in Medicinal Chemistry
Volume: 16 Issue: 3 Year: 2016 Page: 218-226
Author(s): Federica De Angelis,Ada Maria Tata

Exploration of N-arylpiperazine Binding Sites of D2 Dopaminergic Receptor

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 15 Issue: 12 Year: 2015 Page: 988-1001
Author(s): Vukic Soskic,Vladimir Sukalovic,Sladjana Kostic-Rajacic

Pharmacological Approaches to Targeting Muscarinic Acetylcholine Receptors

Journal: Recent Patents on CNS Drug Discovery (Discontinued)
Volume: 9 Issue: 2 Year: 2014 Page: 85-100
Author(s): Carlo Matera, Ada M. Tata

Allosteric Enhancers of A1 Adenosine Receptors: State of the Art and New Horizons for Drug Development

Journal: Current Medicinal Chemistry
Volume: 17 Issue: 3 Year: 2010 Page: 3488-3502
Author(s): R. Romagnoli, P. G. Baraldi, M. A. Tabrizi, S. Gessi, P. A. Borea, S. Merighi

Review Article

Tuning Down the Pain – An Overview of Allosteric Modulation of Opioid Receptors: Mechanisms of Modulation, Allosteric Sites, Modulator Syntheses

Journal: Current Topics in Medicinal Chemistry
Volume: 20 Issue: 31 Year: 2020 Page: 2852-2865
Author(s): Damian Bartuzi,Tomasz M. Wróbel,Agnieszka A. Kaczor,Dariusz Matosiuk

Multifunctional Tacrine Derivatives in Alzheimer’s Disease

Journal: Current Topics in Medicinal Chemistry
Volume: 13 Issue: 1 Year: 2013 Page: 1771-1786
Author(s): Anna Minarini, Andrea Milelli, Elena Simoni, Michela Rosini, Maria Laura Bolognesi, Chiara Marchetti, Vincenzo Tumiatti

Synthesis, Pharmacological Activity and Molecular Modeling of 1-Aryl-7- hydroxy-2,3-dihydroimidazo[1,2-a]pyrimidine-5(1H)-ones and their 6-Substituted Derivatives

Journal: Medicinal Chemistry
Volume: 10 Issue: 5 Year: 2014 Page: 460-475
Author(s): Marzena Rzadkowska,Elzbieta Szacon,Agnieszka A. Kaczor,Sylwia Fidecka,Ewa Kedzierska,Dariusz Matosiuk

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