Search Result "P-gp modulation assays"

A Transcellular Assay to Assess the P-gp Inhibition in Early Stage of Drug Development

Journal: Drug Metabolism Letters
Volume: 6 Issue: 4 Year: 2012 Page: 285-291
Author(s): Jan-Shiang Taur, Edgar L. Schuck, Nancy Y. Wong

Modulation and Absorption of Xenobiotics: The Synergistic Role of CYP450 and P-gp Activities in Cancer and Neurodegenerative Disorders

Journal: Current Drug Metabolism
Volume: 12 Issue: 8 Year: 2011 Page: 702-712
Author(s): Carmela Inglese, Maria Grazia Perrone, Francesco Berardi, Roberto Perrone, Nicola Antonio Colabufo

Recent Developments of P-gp Inhibitors

Ebook: Advances in Anticancer Agents in Medicinal Chemistry
Volume: 1 Year: 2013
Author(s): Sören Krawczyk,Christiane Baumert,Andreas Hilgeroth
Doi: 10.2174/9781608054930113010008

Review Article

Flavonoids as P-gp Inhibitors: A Systematic Review of SARs

Journal: Current Medicinal Chemistry
Volume: 26 Issue: 25 Year: 2019 Page: 4799-4831
Author(s): Jiahua Cui,Xiaoyang Liu,Larry M.C. Chow

Three Decades of P-gp Inhibitors: Skimming Through Several Generations and Scaffolds

Journal: Current Medicinal Chemistry
Volume: 19 Issue: 13 Year: 2012 Page: 1946-2025
Author(s): A. Palmeira,E. Sousa,M. H. Vasconcelos,M. M. Pinto

Evaluating Potential P-gp Substrates: Main Aspects to Choose the Adequate Permeability Model for Assessing Gastrointestinal Drug Absorption

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 15 Issue: 10 Year: 2015 Page: 858-871
Author(s): Joao Batista da Silva Junior,Thaisa Marinho Dezani,Andre Bersani Dezani,Cristina Helena dos Reis Serra

Review Article

Design and Synthesis of New Selective P-gp Substrates and Inhibitors

Journal: Current Pharmaceutical Design
Volume: 22 Issue: 38 Year: 2016 Page: 5774-5778
Author(s): Mariangela Cantore,Marcello Leopoldo,Francesco Berardi,Roberto Perrone,Nicola Antonio Colabufo

11C-verapamil to Assess P-gp Function in Human Brain During Aging,Depression and Neurodegenerative Disease

Journal: Current Topics in Medicinal Chemistry
Volume: 10 Issue: 1 Year: 2010 Page: 1775-1784
Author(s): A. L. Bartels, O. L. de Klerk, R. Kortekaas, J. J. de Vries, K. L. Leenders

Strategies for Targeting the Multidrug Resistance-1 (MDR1)/P-gp Transporter in Human Malignancies

Journal: Current Cancer Drug Targets
Volume: 5 Issue: 6 Year: 2005 Page: 445-455
Author(s): Daruka Mahadevan, Nikhil Shirahatti

Substrates, Inhibitors and Activators of P-glycoprotein: Candidates for Radiolabeling and Imaging Perspectives

Journal: Current Topics in Medicinal Chemistry
Volume: 10 Issue: 1 Year: 2010 Page: 1703-1714
Author(s): Nicola A. Colabufo, Francesco Berardi, Maria Grazia Perrone, Elena Capparelli, Mariangela Cantore, Carmela Inglese, Roberto Perrone

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