Search Result "LEDGF/p75 inhibitor"


Recent Advances in the Development of Small-Molecular Inhibitors Target HIV Integrase-LEDGF/p75 Interaction

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 15 Issue: 14 Year: 2015 Page: 1195-1208
Author(s): Yu Zhao,Zaigang Luo

Research Article

Quantitative Structure-Activity Relationship Study for HIV-1 LEDGF/p75 Inhibitors

Journal: Current Computer-Aided Drug Design
Volume: 16 Issue: 5 Year: 2020 Page: 654-666
Author(s): Yang Li,Yujia Tian,Yao Xi,Zijian Qin,Aixia Yan

Research Article

Quinoline-based Protein–protein Interaction Inhibitors of LEDGF/p75 and HIV Integrase: An In Silico Study

Journal: Current Topics in Medicinal Chemistry
Volume: 18 Issue: 32 Year: 2018 Page: 2800-2815
Author(s): Nisha Chhokar,Sourav Kalra,Monika Chauhan,Anjana Munshi,Raj Kumar

Inhibition of the Interaction between HIV-1 Integrase and its Cofactor LEDGF/p75: A Promising Approach in Anti-Retroviral Therapy

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 11 Issue: 8 Year: 2011 Page: 714-727
Author(s): L. De Luca, S. Ferro, F. Morreale, A. Chimirri

Targeting Virus-host Interactions of HIV Replication

Journal: Current Topics in Medicinal Chemistry
Volume: 16 Issue: 1 Year: 2016 Page: 1167-1190
Author(s): Caroline Weydert, Jan De Rijck, Frauke Christ, Zeger Debyser

Allosteric Integrase Inhibitors

Ebook: Frontiers in Clinical Drug Research: HIV
Volume: 3 Year: 2016
Author(s): Victoria Hann,Peter Dawson,Mark Ashton
Doi: 10.2174/9781681082295116030004

HIV Integrase - Biology and Inhibitor Design

Ebook: Frontiers in Clinical Drug Research: HIV
Volume: 1 Year: 2015
Author(s): Victoria Hann,Mark Ashton
Doi: 10.2174/9781608058969114010008

Mechanisms Governing Lentivirus Integration Site Selection

Journal: Current Gene Therapy
Volume: 8 Issue: 6 Year: 2008 Page: 419-429
Author(s): Angela Ciuffi

Pharmacophore Modelling as a Virtual Screening Tool for the Discovery of Small Molecule Protein-protein Interaction Inhibitors

Journal: Current Pharmaceutical Design
Volume: 18 Issue: 30 Year: 2012 Page: 4586-4598
Author(s): Arnout Voet,Kam Y.J. Zhang

Will Integrase Inhibitors be Used as Microbicides?

Journal: Current HIV Research
Volume: 10 Issue: 1 Year: 2012 Page: 36-41
Author(s): Giuliana C. Crucitti, Maurizio Botta, Roberto Di Santo

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