Search Result "JQ1."
The BET-Bromodomain Inhibitor JQ1 Reduces Inflammation and Tau Phosphorylation at Ser396 in the Brain of the 3xTg Model of Alzheimerâs Disease
Journal: Current Alzheimer Research
Volume: 13 Issue: 9 Year: 2016 Page: 985-995
Author(s): Marco Magistri,Dmitry Velmeshev,Madina Makhmutova,Prutha Patel,Gregory C. Sartor,Claude-Henry Volmar,Claes Wahlestedt,Mohammad Ali Faghihi
The Killing of Human Neuroblastoma Cells by the Small Molecule JQ1 Occurs in a p53-Dependent Manner
Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 20 Issue: 13 Year: 2020 Page: 1613-1625
Author(s): Joseph Mazar,Caleb Gordon,Varun Naga,Tamarah J. Westmoreland
JQ1, a BET Inhibitor, Synergizes with Cisplatin and Induces Apoptosis in Highly Chemoresistant Malignant Pleural Mesothelioma Cells
Journal: Current Cancer Drug Targets
Volume: 18 Issue: 8 Year: 2018 Page: 816-828
Author(s): Ilaria Zanellato,Donato Colangelo,Domenico Osella
An Overview on Small Molecule Inhibitors of BRD4
Journal: Mini-Reviews in Medicinal Chemistry
Volume: 16 Issue: 17 Year: 2016 Page: 1403-1414
Author(s): Wenhai Huang,Xiaoliang Zheng,Yewei Yang,Xiaoju Wang,Zhengrong Shen
The Bromodomain and Extra-Terminal Protein Inhibitor OTX015 Suppresses T Helper Cell Proliferation and Differentiation
Journal: Current Molecular Medicine
Volume: 18 Issue: 9 Year: 2018 Page: 594-601
Author(s): Xiao Hu,Lauren P. Schewitz-Bowers,Philippa J. P. Lait,David A. Copland,Madeleine L. Stimpson,Jing Jing Li,Yizhi Liu,Andrew D. Dick,Richard W. J. Lee,Lai Wei
Designer Benzodiazepinesâ Activity on Opioid Receptors: A Docking Study
Journal: Current Pharmaceutical Design
Volume: 28 Issue: 32 Year: 2022 Page: 2639-2652
Author(s): John Martin Corkery
Drug Discovery of Acetophenone Derivatives as BRD4 Inhibitors
Journal: Letters in Drug Design & Discovery
Volume: 17 Issue: 3 Year: 2020 Page: 323-329
Author(s): Zhimin Zhang,Wenhai Huang,Xiaoliang Zheng,Chuansheng Li,Zhengrong Shen
Dual-target Inhibitors Based on BRD4: Novel Therapeutic Approaches for Cancer
Journal: Current Medicinal Chemistry
Volume: 28 Issue: 9 Year: 2021 Page: 1775-1795
Author(s): Sitao Zhang,Yanzhao Chen,Chengsen Tian,Yujing He,Zeru Tian,Yichao Wan,Tingting Liu
MYC-mediated Synthetic Lethality for Treatment of Hematological Malignancies
Journal: Current Cancer Drug Targets
Volume: 15 Issue: 1 Year: 2015 Page: 53-70
Author(s): Xin Li,Xin A. Zhang,Wei Xie,Xiaoqing Li,Shiang Huang
Recent Developments in Targeting Bromodomain and Extra TerminalDomain Proteins for Cancer Therapeutics
Journal: Current Medicinal Chemistry
Volume: 29 Issue: 25 Year: 2022 Page: 4391-4409
Author(s):