Search Result "Efflux pump inhibitor hybrids"


Efflux Pump Inhibitors: A Novel Approach to Combat Efflux-Mediated Drug Resistance in Bacteria

Journal: Current Drug Targets
Volume: 17 Issue: 6 Year: 2016 Page: 702-719
Author(s): Yinhu Wang, Henrietta Venter, Shutao Ma

Review Article

An Update on Staphylococcus aureus NorA Efflux Pump Inhibitors

Journal: Current Topics in Medicinal Chemistry
Volume: 20 Issue: 24 Year: 2020 Page: 2168-2185
Author(s): Kadja Luana Chagas Monteiro,Thiago Mendonça de Aquino,Francisco Jaime B. Mendonça Junior

Bacterial Resistance Mechanisms and Inhibitors of Multidrug Efflux Pumps Belonging to the Major Facilitator Superfamily of Solute Transport Systems

Ebook: Frontiers in Anti-Infective Drug Discovery
Volume: 5 Year: 2017
Author(s): Manuel F. Varela,Jody L. Andersen,K.C. Ranjana,Sanath Kumar,Leslie M. Sanford,Alberto J. Hernandez
Doi: 10.2174/9781681082912117050006

Review Article

Small Molecule Efflux Pump Inhibitors in Mycobacterium tuberculosis: A Rational Drug Design Perspective

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 18 Issue: 1 Year: 2018 Page: 72-86
Author(s): Erika Kapp,Sarel F. Malan,Jacques Joubert,Samantha L. Sampson

Microbial Efflux Pump Inhibition: Tactics and Strategies

Journal: Current Pharmaceutical Design
Volume: 17 Issue: 1 Year: 2011 Page: 1291-1302
Author(s): George P. Tegos, Mark Haynes, J. Jacob Strouse, Mohiuddin Md. T. Khan, Cristian G. Bologa, Tudor I. Oprea, Larry A. Sklar

Challenges in Oral Delivery: Role of P-gp Efflux Pump

Journal: Current Drug Therapy
Volume: 9 Issue: 1 Year: 2014 Page: 47-55
Author(s): Karan Mittal,Rajashree C. Mashru,Arti R. Thakkar

Research Article

Overexpression of Efflux Pumps AcrAB and OqxAB Contributes toCiprofloxacin Resistance in Clinical Isolates of K. pneumoniae

Journal: Current Protein & Peptide Science
Volume: 23 Issue: 5 Year: 2022 Page: 356-368
Author(s): Melda Meral Öcal

The AcrB Efflux Pump: Conformational Cycling and Peristalsis Lead to Multidrug Resistance

Journal: Current Drug Targets
Volume: 9 Issue: 9 Year: 2008 Page: 729-749
Author(s): Markus A. Seeger, Kay Diederichs, Thomas Eicher, Lorenz Brandstatter, Andre Schiefner, Francois Verrey, Klaas M. Pos

Multidrug Resistance and Efflux Pumps: Insights from Molecular Dynamics Simulations

Journal: Current Topics in Medicinal Chemistry
Volume: 13 Issue: 24 Year: 2013 Page: 3165-3183
Author(s): Francesca Collu,Michele Cascella

Review Article

Transition Towards Antibiotic Hybrid Vehicles: The Next GenerationAntibacterials

Journal: Current Medicinal Chemistry
Volume: 30 Issue: 1 Year: 2023 Page: 104-125
Author(s):

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