Search Result "BRAF <sup>(V600E)</sup> kinase"


Design, Synthesis and Antitumor Activities of Bis-arylureas and Bis-arylamides Based on1H-benzo[d]imidazole Moiety as Novel BRafV600E/VEGFR2 Dual inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 11 Issue: 9 Year: 2014 Page: 1079-1089
Author(s): Weimin Yang,Yadong Chen,Yanmin Zhang,Sanzhi Tang,Hongli Chen,Weifang Tang,Tao Lu

Insight into the Binding of DFG-out Allosteric Inhibitors to B-Raf Kinase Using Molecular Dynamics and Free Energy Calculations

Journal: Current Computer-Aided Drug Design
Volume: 11 Issue: 2 Year: 2015 Page: 124-136
Author(s): Luis Coronel,Jose M. Granadino-Roldán,Marta Pinto,Maria S. Tomas,Maria D. Pujol,Jaime Rubio-Martinez

Ipilimumab and Vemurafenib: Two Different Routes for Targeting Melanoma

Journal: Current Cancer Drug Targets
Volume: 13 Issue: 8 Year: 2013 Page: 879-894
Author(s): Ana Burgeiro,Faustino Mollinedo,Paulo J. Oliveira

Pyrazole Derivatives as Antitumor, Anti-Inflammatory and Antibacterial Agents

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 13 Issue: 13 Year: 2013 Page: 1957-1966
Author(s): Jia-Jia Liu,Meng-yue Zhao,Xin Zhang,Xin Zhao,Hai-Liang Zhu

Research Article

Evaluation of Ligustrazine-Based Synthetic Compounds for their Antiproliferative Effects

Journal: Medicinal Chemistry
Volume: 17 Issue: 9 Year: 2021 Page: 956-962
Author(s): Syed N.A. Bukhari,Nasser H. Alotaibi,Waqas Ahmad,Khalid S. Alharbi,Mohamed A. Abdelgawad,Mohammad M. Al-Sanea,Muhammad M. Ahmad,Muhammad W. Amjad,Maria A.G. Raja,Muhammad A. Hussain

Research Article

Design, Synthesis, and Antiproliferative Activity of Quinazolin-4-One/ChalconeHybrids via the EGFR Inhibition Pathway

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 23 Issue: 17 Year: 2023 Page: 1932-1943
Author(s): Heba A. Hassan,Hesham A. M. Gomaa,Bahaa G.M. Youssif,Alaa M. Hayalah

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