Search Result "BET bromodomain inhibition"


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The BET-Bromodomain Inhibitor JQ1 Reduces Inflammation and Tau Phosphorylation at Ser396 in the Brain of the 3xTg Model of Alzheimer’s Disease

Journal: Current Alzheimer Research
Volume: 13 Issue: 9 Year: 2016 Page: 985-995
Author(s): Marco Magistri,Dmitry Velmeshev,Madina Makhmutova,Prutha Patel,Gregory C. Sartor,Claude-Henry Volmar,Claes Wahlestedt,Mohammad Ali Faghihi

Review Article

BET Inhibitors as Anticancer Agents: A Patent Review

Journal: Recent Patents on Anti-Cancer Drug Discovery
Volume: 12 Issue: 4 Year: 2017 Page: 340-364
Author(s): Imran Ali,Gildon Choi,Kwangho Lee

Research Article

Prediction of Inhibition Activity of BET Bromodomain Inhibitors using Grid Search-Based Extreme Learning Machine and Molecular Docking

Journal: Letters in Drug Design & Discovery
Volume: 18 Issue: 11 Year: 2021 Page: 1039-1049
Author(s): Oluwatoba Emmanuel Oyeneyin,Babatunde Samuel Obadawo,Segun Michael Orimoloye,Eric Oluwafisayo Akintemi,Nureni Ipinloju,Adeola M. Asere,Taoreed O. Owolabi

Small-Molecule BET Inhibitors in Clinical and Preclinical Development and Their Therapeutic Potential

Journal: Current Topics in Medicinal Chemistry
Volume: 15 Issue: 8 Year: 2015 Page: 776-794
Author(s): Lei Yu,Zhen Wang,Zhang Zhang,Xiaomei Ren,Xiaoyun Lu,Ke Ding

Review Article

Aim for the Readers! Bromodomains As New Targets Against Chagas’ Disease

Journal: Current Medicinal Chemistry
Volume: 26 Issue: 3 Year: 2019 Page: 6544-6563
Author(s): Victoria Lucia Alonso,Luis Emilio Tavernelli,Alejandro Pezza,Pamela Cribb,Carla Ritagliati,Esteban Serra

Review Article

Privileged Scaffolds Targeting Bromodomain-containing Protein 4

Journal: Current Topics in Medicinal Chemistry
Volume: 22 Issue: 7 Year: 2022 Page: 600-627
Author(s):

Research Article

Overexpression of Bromodomain and Extraterminal Domain is Associated withProgression, Metastasis and Unfavorable Outcomes: Highlighting Prognostic andTherapeutic Value of the BET Protein Family in Gastric Cancer

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 23 Issue: 7 Year: 2023 Page: 794-806
Author(s): Shahrzad S. Fard,Seyed A. Mousavi,Seyed H. Ghaffari

Review Article

Recent Advances in the Development of CBP/p300 Bromodomain Inhibitors

Journal: Current Medicinal Chemistry
Volume: 27 Issue: 33 Year: 2020 Page: 5583-5598
Author(s): Ying Xiong,Mingming Zhang,Yingxia Li

Research Article

Synthesis and Biological Activity of Quinoxalone Derivatives as BRD4 Bromodomain Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 1 Year: 2017 Page: 50-57
Author(s): Bin Xu,Lei-Lei Zhao,Yi-Fei Yang,Jian Zhang,Ling-Yun Yang,Bing Zhang,Li Han,Hui-Bin Zhang,Jin-Pei Zhou

Review Article

Recent Developments in Targeting Bromodomain and Extra TerminalDomain Proteins for Cancer Therapeutics

Journal: Current Medicinal Chemistry
Volume: 29 Issue: 25 Year: 2022 Page: 4391-4409
Author(s):

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