Search Result "β-secretase (BACE-1)"


2D QSAR Studies on Series of Human Beta-secretase (BACE-1) Inhibitors

Journal: Medicinal Chemistry
Volume: 10 Issue: 2 Year: 2014 Page: 162-173
Author(s): Daniela Santos Cruz, Marcelo Santos Castilho

Progress in the Development of Nonpeptidomimetic BACE 1 Inhibitors for Alzheimers Disease

Journal: Current Medicinal Chemistry
Volume: 16 Issue: 1 Year: 2009 Page: 1806-1820
Author(s): Wen-Hai Huang, Rong Sheng, Yong-Zhou Hu

Beta-Secretase: Structure, Function, and Evolution

Journal: CNS & Neurological Disorders - Drug Targets
Volume: 7 Issue: 3 Year: 2008 Page: 278-294
Author(s): Chitra Venugopal, Christina M. Demos, K. S. Jagannatha Rao, Miguel A. Pappolla, Kumar Sambamurti

Review of Synthesis, Assay, and Prediction of β and γ-secretase Inhibitors

Journal: Current Topics in Medicinal Chemistry
Volume: 12 Issue: 8 Year: 2012 Page: 828-844
Author(s): Helena Nino,Jose Enrique Rodriguez-Borges,Xerardo Garcia-Mera,Francisco Prado-Prado

Research Article

Pharmacophore Modeling and Docking Studies to Investigate Potential Leads for the Development of β -Secretase APP Cleavage Enzyme-1 (BACE-1) Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 16 Issue: 7 Year: 2019 Page: 775-784
Author(s): Richa Arya,Satya Prakash Gupta,Sarvesh Paliwal,Swapnil Sharma,Kirtika Madan,Monika Chauhan

Short Communication

Exploring the Molecular Structural Requirements of Flavonoids as Beta-Secretase-1 Inhibitors Using Molecular Modeling Studies

Journal: Current Drug Discovery Technologies
Volume: 20 Issue: 3 Year: 2023 Page: 52-65
Author(s): Uttam A. More,Malleshappa N. Noolvi

Review Article

Dual BACE-1/GSK-3β Inhibitors to Combat Alzheimer's Disease: A Focused Review

Journal: Current Topics in Medicinal Chemistry
Volume: 17 Issue: 31 Year: 2017 Page: 3361-3369
Author(s): Angela Rampa,Silvia Gobbi,Rita Maria Concetta Di Martino,Federica Belluti,Alessandra Bisi

Research Article

QSAR and Molecular Modeling Studies on a Series of Pyrrolidine Analogs Acting as BACE-1 Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 16 Issue: 7 Year: 2019 Page: 746-760
Author(s): Richa Arya,Satya Prakash Gupta,Sarvesh Paliwal,Seema Kesar,Achal Mishra,Yenamandra Subrahmanya Prabhakar

Design of Some New Potent Beta-secretase Inhibitors Based on QSAR and Molecular Modeling Study on a Series of Hydroxyethylamine Derivatives

Journal: Letters in Drug Design & Discovery
Volume: 10 Issue: 3 Year: 2013 Page: 253-265
Author(s): YashShree Pandey,Satya Prakash Gupta

Memapsin 2 (Beta-Secretase) Inhibitors: Drug Development

Journal: Current Alzheimer Research
Volume: 5 Issue: 2 Year: 2008 Page: 121-131
Author(s): Arun K. Ghosh, Nagaswamy Kumaragurubaran, Ling Hong, Gerald Koelsh, Jordan Tang

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