[1]
Kim, B.M.; Williams, S.F.; Masamune, S. In: Comprehensive Organic Synthesis; Trost, B.M.; Fleming, I.; Heathcock, C.H., Eds.; Pergamon: Oxford, 1991, Vol. 2, pp. 229-275.
[2]
Eder, U.; Sauer, G.; Wiechert, R. New type of asymmetric cyclization to optically active steroid CD partial structures. Angew. Chem. Int. Ed. Engl., 1971, 10, 496-497.
[3]
Hajos, Z.G.; Parrish, D.R. Asymmetric synthesis of bicyclic intermediates of natural product chemistry. J. Org. Chem., 1974, 39, 1615-1621.
[4]
List, B.; Lerner, R.A.; Barbas III, C.F. Proline-catalyzed direct asymmetric aldol reactions. J. Am. Chem. Soc., 2000, 122, 2395-2396.
[5]
Ahrendt, K.A.; Borths, C.J.; MacMillan, D.W.C. New strategies for organic catalysis: the first highly enantioselective organocatalytic Diels−Alder reaction. J. Am. Chem. Soc., 2000, 122, 4243-4244.
[6]
Enantioselective Organocatalysis, Reactions and Experimental
Procedures;; Dalko, P.I. Ed.; Wiley-VCH: Weinheim,. , 2007.
[7]
Asymmetric Organocatalysis, From Biomimetic Concepts to Applications
in Asymmetric Synthesis;; Berkessel, A.; Gröger, H. Eds.;
Wiley-VCH: Weinheim,. , 2005.
[8]
Comprehensive Enantioselective Organocatalysis: Catalysts, Reactions, and Applications; Dalko, P.I. Ed.; Wiley-VCH: Weinheim,. , 2013.
[9]
Notz, W.; List, B. Catalytic asymmetric synthesis of anti-1,2-diols. J. Am. Chem. Soc., 2000, 122, 7386-7387.
[10]
Sakthivel, K.; Notz, W.; Bui, T.; Barbas III, C.F. Amino acid catalyzed direct asymmetric aldol reactions: A bioorganic approach to catalytic asymmetric carbon-carbon bond-forming reactions. J. Am. Chem. Soc., 2001, 123, 5260-5267.
[11]
List, B. Enamine catalysis is a powerful strategy for the catalytic generation and use of carbanion equivalents. Acc. Chem. Res., 2004, 37, 548-557.
[12]
Notz, W.; Tanaka, F.; Barbas III, C.F. Enamine-based organocatalysis with proline and diamines: The development of direct catalytic asymmetric aldol, Mannich, Michael, and Diels-Alder Reactions. Acc. Chem. Res., 2004, 37, 580-591.
[13]
List, B. Proline-catalyzed asymmetric reactions. Tetrahedron, 2002, 58, 5573-5590.
[14]
Bisai, V.; Bisai, A.; Singh, V.K. Enantioselective organocatalytic aldol reaction using small organic molecules. Tetrahedron, 2012, 68, 4541-4580.
[15]
Trost, B.M.; Brindle, C.S. The direct catalytic asymmetric aldol reaction. Chem. Soc. Rev., 2010, 39, 1600-1632.
[16]
Pellissier, H. Asymmetric organocatalysis. Tetrahedron, 2007, 63, 9267-9331.
[17]
Guillena, G. Organocatalyzed aldol reactions. In: Modern Methods in Stereoselective Aldol Reactions; Mahrwald, R., Ed.; Wiley-VCH: Weinheim, 2013, pp. 155-268.
[18]
Heravi, M.M.; Zadsirjan, V.; Dehghani, M.; Hosseintash, N. Current applications of organocatalysts in asymmetric aldol reactions: An update. Tetrahedron Asymmetry, 2017, 28, 587-707.
[19]
Tang, Z.; Jiang, F.; Yu, L-T.; Gong, L-Z.; Mi, A-Q.; Jiang, Y-Z.; Wu, Y-D. Novel small organic molecules for a highly enantioselective direct aldol reaction. J. Am. Chem. Soc., 2003, 125, 5262-5263.
[20]
Tang, Z.; Jiang, F.; Cui, X.; Gong, L-Z.; Mi, A-Q.; Jiang, Y-Z.; Wu, Y-D. Enantioselective direct aldol reactions catalyzed by L-prolinamide derivatives. Proc. Natl. Acad. Sci. USA, 2004, 101, 5755-5760.
[21]
Tang, Z.; Yang, Z-H.; Chen, X-H.; Cun, L-F.; Mi, A-Q.; Jiang, Y-Z.; Gong, L-Z. A highly efficient organocatalyst for direct aldol reactions of ketones with aldedydes. J. Am. Chem. Soc., 2005, 127, 9285-9289.
[22]
Samanta, S.; Liu, J.; Dodda, R.; Zhao, C-G. C2-symmetric bisprolinamide as a highly efficient catalyst for direct aldol reaction. Org. Lett., 2005, 7, 5321-5323.
[23]
Chen, J-R.; Lu, H-H.; Li, X-Y.; Chen, L.; Wan, J.; Xiao, W-J. Readily tunable and bifunctional L-prolinamide derivatives: Design and application in the direct enantioselective aldol reactions. Org. Lett., 2005, 7, 4543-4545.
[24]
Chen, J-R.; Li, X-Y.; Xing, X-N.; Xiao, W-J. Sterically and electronically tunable and bifunctional organocatalysts: Design and application in asymmetric aldol reaction of cyclic ketones with aldehydes. J. Org. Chem., 2006, 71, 8198-8202.
[25]
Chen, J-R.; An, X-L.; Zhu, X-Y.; Wang, X-F.; Xiao, W-J. Rational combination of two privileged chiral backbones: Highly efficient organocatalysts for asymmetric direct aldol reactions between aromatic aldehydes and acylic ketones. J. Org. Chem., 2008, 73, 6006-6009.
[26]
Gandhi, S.; Singh, V.K. Synthesis of chiral organocatalysts derived from aziridines: Application in asymmetric aldol reaction. J. Org. Chem., 2008, 73, 9411-9416.
[27]
Rojas Cabrera, H.; Huelgas, G.; Hernandez Perez, J.M.; Walsh, P.J.; Somanathan, R.; Anaya de Parrodi, C. Homochiral L-prolinamido-sulfonamides and their use as organocatalysts in aldol reactions. Tetrahedron Asymmetry, 2015, 26, 163-172.
[28]
Kucherenko, A.S.; Syutkin, D.E.; Zlotin, S.G. Asymmetric aldol condensation in an ionic liquid-water system catalyzed by (S)-prolinamide derivatives. Russ. Chem. Bull. Int. Ed., 2008, 57, 59-594.
[29]
Chen, F.; Huang, S.; Zhang, H.; Liu, F.; Peng, Y. Proline-based dipeptides with two amide units as organocatalyst for the asymmetric aldol reaction of cyclohexanone with aldehydes. Tetrahedron, 2008, 64, 9585-9591.
[30]
Maleev, V.I.; Gugkaeva, Z.T.; Moskalenko, M.A.; Tsaloev, A.T.; Lyssenko, K.A. New (S)-proline derivatives as catalysts for the enantioselective aldol reaction. Russ. Chem. Bull. Int. Ed, 2009, 58, 1903-1907.
[31]
De Nisco, M.; Pedatella, S.; Ullah, H.; Zaidi, J.H.; Naviglio, D.; Özdamar, O.; Caputo, R. Proline−β3-amino-ester dipeptides as efficient catalysts for enantioselective direct aldol reaction in aqueous medium. J. Org. Chem., 2009, 74, 9562-9565.
[32]
Tzeng, Z-H.; Chen, H-Y.; Reddy, R-J.; Huang, C-T.; Chen, K. Highly diastereo- and enantioselective direct aldol reactions promoted by water-compatible organocatalysts bearing a pyrrolidinyl-camphor structural scaffold. Tetrahedron, 2009, 65, 2879-2888.
[33]
Yang, Y.; He, Y-H.; Guan, Z.; Huang, W-D. A highly efficient large-scale asymmetric direct intermolecular aldol reaction employing L-prolinamide as a recoverable catalyst. Adv. Synth. Catal., 2010, 352, 2579-2587.
[34]
Saha, S.; Moorthy, J.N. Highly enantioselective aldol reactions using N-arylprolinamides with enhanced acidity and double H-bonding potential. Tetrahedron Lett., 2010, 51, 912-916.
[35]
Subba Reddy, B.V.; Bhavani, K.; Raju, A.; Yadav, J.S. A novel trifunctional organocatalyst for the asymmetric aldol reaction: a facile enantioselective synthesis of β-hydroxyketones. Tetrahedron Asymmetry, 2011, 22, 881-886.
[36]
Hernández, J.G.; García-López, V.; Juaristi, E. Solvent-free asymmetric aldol reaction organocatalyzed by (S)-proline-containing thiodipeptides under ball-milling conditions.-. Tetrahedron, 2012, 68, 92-97.
[37]
Sutar, R.L.; Joshi, N.N. Systematic evaluation of a few proline derivatives as catalysts for a direct aldol reaction. Tetrahedron Asymmetry, 2013, 24, 43-49.
[38]
Bañón-Caballero, A.; Guillena, G.; Nájera, C.; Faggi, E.; Sebastián, R.M.; Vallribera, A. Recoverable silica-gel supported binam-prolinamides as organocatalysts for the enantioselective solvent-free intra- and intermolecular aldol reaction. Tetrahedron, 2013, 69, 1307-1315.
[39]
Pedrosa, R.; Andrés, J.M.; Gamarra, A.; Manzano, R.; Pérez-López, C. Novel sulfonylpolystyrene-supported prolinamides as catalysts for enantioselective aldol reaction in water. Tetrahedron, 2013, 69, 10811-10819.
[40]
Samanta, S.; Zhao, C-G. Asymmetric direct aldol reaction of 1,2-diketones and ketones mediated by proline derivatives. Tetrahedron Lett., 2006, 47, 3383-3386.
[41]
Mitchell, J.M.; Finney, N.S. An efficient method for the preparation of N, N-disubstituted 1, 2-diamines. Tetrahedron Lett., 2000, 41, 8431-8434.
[42]
Xu, D.; Prasad, K.; Repic, O.; Blacklock, T.J. Ethyl trifluoroacetate: a powerful reagent for differentiating amino groups. Tetrahedron Lett., 1995, 36, 7357-7360.
[43]
Manville, C.V.; Docherty, G.; Padda, R.; Wills, M. Application of proline-functionalized 1,2-diphenylethane-1,2-diamine (DPEN) in asymmetric transfer hydrogenation of ketones. Eur. J. Org. Chem., 2011, 6893-6901.
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