Abstract
This review reports the chemistry of 2,3-disubstituted N-H aziridines to Five and sixmemberd N-heterocycles. Emphasis will be put on the aspects of stereo- and regioselectivity of appropriate reactions such as 1,3-dipolar, ring expansion reactions as well as C-C or C-N bond cleavage of aziridine ring.
Keywords: Ketoaziridine, rearrangement, ring expansion, stereo- and regioselectivity.
Graphical Abstract
Mini-Reviews in Organic Chemistry
Title:Ring Expansion of N-H Ketoaziridines to Five and Six-Membered NHeterocycles
Volume: 12 Issue: 4
Author(s): Heshmat A. Samimi
Affiliation:
Keywords: Ketoaziridine, rearrangement, ring expansion, stereo- and regioselectivity.
Abstract: This review reports the chemistry of 2,3-disubstituted N-H aziridines to Five and sixmemberd N-heterocycles. Emphasis will be put on the aspects of stereo- and regioselectivity of appropriate reactions such as 1,3-dipolar, ring expansion reactions as well as C-C or C-N bond cleavage of aziridine ring.
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Cite this article as:
Samimi A. Heshmat, Ring Expansion of N-H Ketoaziridines to Five and Six-Membered NHeterocycles, Mini-Reviews in Organic Chemistry 2015; 12 (4) . https://dx.doi.org/10.2174/1570193X12666150930224129
DOI https://dx.doi.org/10.2174/1570193X12666150930224129 |
Print ISSN 1570-193X |
Publisher Name Bentham Science Publisher |
Online ISSN 1875-6298 |
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