First Efficient One-Pot Synthesis of Tetrahydropyrrolo[2,3-d]azocines and Tetrahydroazocino[4,5-b]indoles

Title: First Efficient One-Pot Synthesis of Tetrahydropyrrolo[2,3-d]azocines and Tetrahydroazocino[4,5-b]indoles

Volume: 2 Issue: 1

Author(s): Leonid G. Voskressensky, Tatiana N. Borisova, Tatiana A. Soklakova, Larisa N. Kulikova, Roman S. Borisov and Alexej V. Varlamov

Affiliation:

Keywords: ring expansion, tandem cleavage, azocines, pyrroles, carbolines

Abstract: A new efficient one-pot protocol for the synthesis of tetrahydropyrrolo[2,3-d]azocines and tetrahydroazocino[4,5-b]indoles starting from ready-available tetrahydropyrrolo[3,2-c]pyridines and tetrahydropyrido[4,3-b]indoles correspondingly and dimethylacetylene dicarboxylate or ethyl propiolate is being offered.

Cite this article as:

Voskressensky G. Leonid, Borisova N. Tatiana, Soklakova A. Tatiana, Kulikova N. Larisa, Borisov S. Roman and Varlamov V. Alexej, First Efficient One-Pot Synthesis of Tetrahydropyrrolo[2,3-d]azocines and Tetrahydroazocino[4,5-b]indoles, Letters in Organic Chemistry 2005; 2 (1) . https://dx.doi.org/10.2174/1570178053400090